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OLYMPIC

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  1. Clomid (Clomiphene Citrate) is a powerfully effective anti-estrogen officially classified as a Selective Estrogen Receptor Modulator (SERM). In many ways, it is very similar to another popular SERM in Nolvadex (Tamoxifen Citrate). Clomid first gained worldwide attention in the early 1970’s as a strong fertility aid and is still used for that purpose today. It is also one of the most commonly used SERM’s by anabolic steroid users. No, it is not an anabolic steroid but can be used to combat estrogenic side effects sometimes caused by anabolic steroids. It can also be used as a Post Cycle Therapy (PCT) medication in order to stimulate suppressed testosteroneproduction due to anabolic steroid use. PCT use of Clomid is the most common purpose and most beneficial point of use for the anabolic steroid user. Clomid Functions & Traits: Clomiphene Citrate is a SERM that is specifically used as a fertility aid due to its ability to enhance the release of gonadotropins. Clomid has the ability to oppose the negative feedback of estrogens on the Hypothalamic-Pituitary-Ovarian-Axis. This will increase the release of Luteinizing Hormone (LH) and Follicle Stimulating Hormone (FSH) significantly. By increasing gonadotropin release, this can lead to the egg being released, thereby increasing the chance of conception. Clomid also carries strong anti-estrogen properties that could be used therapeutically, but its anti-estrogen properties are most commonly associated with anabolic steroid use. Testosterone and many testosterone derived steroids have the ability to convert to estrogen through testosterone’s interaction with the aromatase enzyme. As estrogen levels rise, this can lead to gynecomastia and excess water retention. Heavy water retention can also promote high blood pressure. By supplementing with Clomid during anabolic steroid use, the SERM will bind to the estrogen receptors, therefore inhibiting the estrogen hormone from binding. This can be very useful in combating gynecomastia, as when Clomid binds to the receptor it prevents estrogen from stimulating the mammary tissue. It can also have a positive impact on water retention, but as it won’t actively reduce serum estrogen levels it’s sometimes not enough. Clomid also possess functioning traits that are beneficial to the anabolic steroid user post anabolic steroid use. Specifically we’re referring to Post Cycle Therapy (PCT). In men, Clomid also has the ability to stimulate the pituitary to release more LH and FSH, which will in turn stimulate enhanced natural testosterone production. This is extremely beneficial to the anabolic steroid user post cycle as natural testosterone levels will be very low due to suppression caused by anabolic steroid use. Effects of Clomid: In a therapeutic setting as a fertility aid, the effects of Clomid are simple. The woman is having difficulty becoming pregnant, Clomid enhances the chance of conception and pregnancy occurs. It doesn’t always work and we’ll look at the process in the administration section, but it will greatly increase the odds of conception and is fairly successful. As an anti-estrogen for on cycle steroid use, Clomid is fairly effective at staving off gynecomastia. It will not reduce estrogen levels or inhibit the aromatization process, but in many cases, binding to the receptors is enough protection for many men. In fact, while there are stronger protective agents, many men would be surprised as to how well a SERM like Clomid can work if they would give it a chance. More importantly, when using Clomid for this purpose it can also have a positive impact on cholesterol levels. While an anti-estrogen, Clomid actually acts as estrogen in the liver, which in turn will promote healthier cholesterol levels. This can be very beneficial to the anabolic steroid user as anabolic steroid use is notorious for promoting unhealthy cholesterol levels. For many men, especially hardcore anabolic steroid users, Clomid is not enough for estrogenic protection. In this case, an Aromatase Inhibitor (AI) like Arimidex (Anastrozole) or Femara (Letrozole) will be needed. AI’s actively inhibit the aromatase process and will see serum estrogen levels reduced. By far they are the most effective at combating gynecomastia and will have more success in combating water retention. In fact, SERM’s like Clomid often do very little to combat water retention. However, in many cases, many performance athletes would do a better job controlling water retention if they did a better job controlling their diet. In off-season bulking plans this requires excess calories to grow. However, many take it too far, especially carbohydrate consumptions, and this will cause you to hold water with or without anabolic steroid use. Add in aromatizing steroids to the equation and water retention will be even greater. Further, AI’s while effective will have a negative impact on cholesterol, which leads us to only one sane conclusion. Control your diet and if you can control gynecomastia with a SERM like Clomid it should be your first choice. Then we’re left with the effects of Clomid as they pertain to PCT. When we supplement with anabolic steroids, this will suppress natural testosterone production. The rate of suppression will be dependent on the steroids being used and to a degree the total dosing, but it will generally be substantial. For this reason, most men will always include exogenous testosterone in their steroid cycles. In fact, it’s not uncommon for it to be the only steroid used. This will protect the individual from a low testosterone condition while on cycle. Unfortunately, once steroid use comes to an end natural testosterone levels will be very low. Natural testosterone production will begin again on its own, but it will take a significant amount of time for levels to reach their previous high state. In fact, total recovery can take months to even a year. Further, natural testosterone recovery is dependent on no prior low testosterone condition existing and assumes that no severe damage was done to the Hypothalamic-Pituitary-Testicular-Axis (HPTA) through improper anabolic steroid use. Due to natural testosterone levels being low post cycle, most men are encouraged to implement a PCT program. This will stimulate natural testosterone production greatly and shorten the total recovery time. It will not return your levels to normal on its own; there is no PCT plan on earth that can do this. However, a solid PCT plan will ensure you have enough testosterone for proper bodily function while your levels continue to naturally rise. Clomid is an excellent choice for this purpose and one of the most commonly used PCT medications. Highly successful PCT programs will often include Clomid and Nolvadex as well as the powerful peptide hormone HCG (Human Chorionic Gonadotropin). Those who forgo Clomid therapy post cycle or any type of PCT plan and are going to be off cycle for an extended period of time will rest in a low testosterone condition for an extended period of time. Not only is this an extremely unhealthy state, it can come with all the traditional low testosterone symptoms. Many will find cortisol levels greatly increase as testosterone levels are low, and as a result, body fat levels go up and strength and muscle mass decrease. If you’re going to be off cycle for an extended period of time, 8 weeks or more there is no reason for forgoing a PCT program. If you are going to be off cycle for less than 8 weeks or bridging with a low dose of exogenous testosterone, which is very common in hardcore bodybuilding circles, this is the only time a PCT would be counterproductive. Side Effects of Clomid: Clomid is one of the most well-tolerated SERM’s and anti-estrogens on the market, and this applies to both men and women. While it carries a very high threshold of toleration, side effects of Clomid do exist and are possible. However, “possible” is the key word and a very important one. Anytime anabolic steroids are discussed as well as non-steroidal items used by anabolic steroid users, many seem to enjoy implying side effects are assured. This is not the case; in fact, most should be able to use Clomid side effect free. When it comes to the possible side effects of Clomid, we will find most are fairly rare. Some women who have used the SERM as a fertility aid have experienced ovarian enlargement, but again this is very rare. Other possible side effects of Clomid use include: Headaches Nausea Hot Flashes Uterine Bleeding (extremely rare) Breast Discomfort The side effects of Clomid are also well noted for including possible visual disturbances. Data shows that approximately 1.5% of all those who use Clomid may experience some type of visual disturbance normally in the form of blurred or hazy vision. If this occurs, use should be discontinued and alternative medications should be examined. In most all cases, once use is discontinued vision will shortly return to normal. However, there have been a few reported cases over the years of visual disturbances that did not remedy post discontinuation. Normally, such cases have been linked to long term and extremely high dose use. Again, if visual disturbances occur, discontinue use immediately and choose another SERM to meet your needs. A final note on the side effects of Clomid, some may experience acne. This appears to be most common when the SERM is used as part of a PCT program. In this case, it’s not really the SERM that’s causing the issue but rather the high influx of natural testosterone that is now being produced. Most should not have an issue, but those who are already genetically sensitive to acne may find a few pimples appear on their back, shoulders or chest. Clomid Administration: For the purpose of fertility aid, Clomid doses will normally be at 50mg per day. The process is very simple; five days into the menstrual cycle a daily 50mg dose is administered every day once a day for five straight days. If this doesn’t result in conception, the dose is sometimes increased to 100mg per day. This cycle will be repeated 5-6 times over the course of the woman’s menstrual cycles until pregnant. If conception does not occur after 5-6 cycles of therapy, alternative treatments will need to be examined. For the anabolic steroid user, standard Clomid doses for on cycle estrogenic protection will normally be 50mg per day throughout the duration of the cycle. If this doesn’t do the trick it’s unlikely any amount of Clomid will work. If this does not provide the protection you need, keep in mind many have reported greater success with the SERM Nolvadex for on cycle protection. However, you may very well need an AI like Arimidex. Then we’re left with PCT Clomid use. Standard PCT Clomid doses will normally start at 100-150mg per day for 1-2 weeks. From here the dose will drop to 50-100mg per day for 1-2 weeks and finish with 1-2 weeks at 50mg per day. Total Clomid therapy should last 4-6 weeks, so dosing should be based and considered on that total schedule. Most will also be far more successful in their PCT recovery by including Nolvadex and HCG. Timing is also important when planning your Clomid PCT use, and this timing factor will vary depending on the inclusion of HCG: If your cycle ends with any large ester base anabolic steroids, you will begin Clomid 2 weeks after your last injection. If your cycle ends with all small ester base anabolic steroids, you will begin your Clomid 3 days after your last injection. If your cycle ends with any large ester base anabolic steroids, you will begin HCG ten days after your last injection and begin Clomid after HCG therapy is complete. If your cycle ends with all small ester base anabolic steroids, you will begin HCG 3 days after your last injection and begin Clomid after HCG therapy is complete. Availability of Clomid: Clomid is available worldwide on both the pharmaceutical and black markets. This is a very easy item to purchase, very affordable and should not be hard to find. In the U.S. it is not a controlled substance, but you will need a prescription to legally buy it. The exception would be a purchase through a research chemical lab (RCL). Numerous RCL’s have popped up over the years providing SERM’s, AI’s, peptides and a host of other items that are not controlled yet require a prescription. By providing such items in their liquid state and for research only, individuals can legally buy them without a prescription. It’s definitely a loophole in the law and it’s one that may not always be there, but it is for now. It is important, however, that you understand the purchase must be for research only. If law enforcement chose to make an issue over it and could prove your purchase was not for research you might find yourself in hot water. Beyond RCL’s, prescription Clomid is not too difficult to get and most black market steroid suppliers carry the SERM. However, if you make a purchase from a steroid supplier, even if you’re not actually buying steroids you will be breaking the law. Buy Clomid Online - Warning: You will find you can easily buy Clomid online from both steroid suppliers and RCL’s and you will find it is very cheap. You will find Clomid tablets are rarely counterfeited, but again you have the legality issue that surrounds such a purchase to contend with. As for an RCL purchase, if you buy Clomid online from an RCL you can easily get a great product. However, as is with underground steroid labs there are more poor RCL’s than quality. Things like under-dosing can be a concern, but more common is an unstable product. Another possible issue is one that’s difficult to dose due to its heavy concentration. Without question, while it is tempting to buy Clomid online your best bet will always be to get the SERM’s or related items you need legally and with a prescription. By obtaining a low testosterone prescription you can easily obtain all the items you need. You may not receive a Clomid prescription, but you will receive all necessary ancillaries. For this reason, for quality and assurance of your legal safety you are encouraged to visit Lowtestosterone.com. Clomid Reviews: Clomid is an excellent SERM and for years there has been an ongoing debate among anabolic steroid users as to which SERM is better, Clomid or Nolvadex. For the purpose of on cycle gynecomastia protection either one can work. Some have reported that Nolvadex tends to do a better job, but you may need to try both at different times to make an accurate assessment. Then we have PCT use, and both are equally effective and important. Many loudly claim Nolvadex is a far superior SERM for PCT purposes; however, there is a common problem with this statement. Most who use Clomid don’t use enough. On a milligram for milligram basis Nolvadex is stronger, so if you don’t plan a Clomid dose to match Nolvadex you’re going to be disappointed in the Clomid. Learn and understand the SERM’s and various items before you use them. Understand proper dosing protocols and you’ll get the most out of Clomid and any SERM you use.
  2. Exemestane is a steroidal Aromatase Inhibitor (AI) that is most commonly known as Aromasin. In fact, the Aromasin brand name is the only pharmaceutical grade brand of the Exemestane AI due to the tight patent Upjohn has maintained on the product. While tightly controlled by the pharmaceutical giant, Aromasin is available in numerous countries around the globe. Aromasin was first released on the U.S. market in 2000 after shortly gaining FDA approval a few months prior in 1999. The primary purpose of use as with most AI’s would be to combat breast cancer in post-menopausal women. Shortly after, the AI would begin to gain a lot of popularity among anabolic steroid users for its ability to protect against estrogenic related side effects. This action is very similar to the older and more popular AI’s in Arimidex (Anastrozole) and Femara (Letrozole). It would also gain a fair amount of popularity in Post Cycle Therapy (PCT) plans among steroid users. It was not the first AI to gain such popularity but would prove to be a little more advantageous for this purpose than most AI’s. Aromasin Functions & Traits: Aromasin is officially classified as a steroidal suicide Aromatase Inhibitor, and carries the ability to inhibit the aromatase enzyme, which is responsible for the production or conversion of testosterone to estrogen. Aromasin has the ability to block aromatization, which in turn inhibits the production of estrogen, and thereby lowers the body’s serum estrogen levels. This will prove useful to breast cancer patients as breast cancer often feeds off the estrogen hormone. It will also prove useful to the anabolic steroid user. Many anabolic steroids have the ability to increase estrogen levels due to the aromatase process, specifically the conversion of testosterone to estrogen. This can lead to gynecomastia and water retention. Excess water retention can also promote high blood pressure when it becomes severe. Steroids that do not carry a strong estrogenic nature can also cause these effects, most notably gynecomastia if they carry a progestin nature. A prime example would be Nandrolone, which while it aromatizes only does so at 20% the rate of testosterone. However, it also carries a strong progestin nature, and progesterone has been well noted for carrying the ability to stimulate the estrogenic mechanism in the mammary tissue. By administering Aromasin during the use of anabolic steroids, this will inhibit the aromatase process, lower estrogen levels and protect the individual from estrogenic side effects. How effective is Aromasin? The product claims on average to have the ability to lower serum estrogen levels by 85%. Aromasin also has the ability to stimulate natural testosterone production, which is precisely why some will include it during their PCT. Like Arimidex and Letrozole, Aromasin will stimulate the pituitary to release more Luteinizing Hormone (LH) and Follicle Stimulating Hormone (FSH), two hormones essential to natural testosterone production. While the other common AI’s share this trait, Aromasin has been shown to carry a slight androgenic effect, as well as the ability to increase the production of Insulin-Like Growth Factor-1 (IGF-1). This is a trait no other AI can claim to carry. By using Aromasin during PCT, the individual receives the desired testosterone boost necessary for recovery, but with the IGF-1 increase also creates a stronger anabolic atmosphere. This is deemed useful by some steroid users as it could potentially give them the ability to protect their lean tissue all the more during use. However, when we look at the direct effects of Aromasin as it pertains to PCT, we will find PCT use is normally not recommended despite these positive effects. Effects of Aromasin: In a therapeutic setting, by blocking the aromatase enzyme, Aromasin actively prohibits the cancer from feeding off the hormone necessary to its survival. It has been proven highly effective for this purpose, but only after the use of the Selective Estrogen Receptor Modulator (SERM) Nolvadex (Tamoxifen Citrate) has failed. While effective, it is also not as commonly used as Arimidex for this purpose as Arimidex largely maintains itself as the primary AI in breast cancer treatment not only among post-menopausal women but in a host of breast cancer scenarios. Then we have Aromasin as an anti-estrogen for the anabolic steroid user. By understanding its functions and traits you should already understand the effects of Aromasin in this regard. Excess estrogen levels can promote gynecomastia and water retention and possibly high blood pressure as a secondary issue. However, keep in mind such effects are not possible with all anabolic steroids, primarily it must carry an estrogenic nature, it must be able to aromatize to lead to such effects or carry a progesterone nature. Testosterone is the primary aromatizing steroid, but testosterone derived steroids like Dianabol can also promote strong estrogenic action. Then we have the Boldenone (Equipoise) hormone, and while it only aromatizes at 50% the rate of testosterone, this is still enough to cause an estrogen buildup in some. Finally, we’re left with 19-nortestosterone (19-nor) anabolic steroids. 19-nor compounds will primarily include all forms of Nandrolone and Trenbolone. As discussed Nandrolone aromatizes at 20% the rate of testosterone, but it also carries a very strong progestin nature. This can promote a fair amount of estrogenic activity in many men. As for Trenbolone, it does not aromatize at all, but its moderately strong progestin nature can make gynecomastia a possibility depending on the individual’s sensitivity. When use is coupled with an aromatizing steroid, this will greatly enhance the odds of gynecomastia. Regardless of the steroid in question, Aromasin can offer protection from the estrogenic effects. An important note: Aromasin will have no affect on dihydrotestosterone (DHT) derived anabolic steroids as they do not convert to estrogen. Such steroids cannot lead to gynecomastia or excess water retention; it is impossible. The exception would be Anadrol (Oxymetholone), while a DHT derivative, it carries with it a strong estrogenic nature. However, while estrogenic action is present, the hormone does not aromatize, meaning there is no aromatization for Aromasin to inhibit. The use of an AI will not affect the estrogenicity of Anadrol. For protection from such a steroid, the individual will need to inhibit activation of the estrogenic mechanism, and this will make SERM’s the first line of defense. The final effects of Aromasin surround its use in a PCT plan. Due to the use of anabolic steroids natural testosterone production is suppressed. The rate of suppression will be dependent on the steroids being used, and to a degree, the total doses, but natural production will be suppressed nonetheless. Most male steroid users are advised to include exogenous testosterone in all their cycles in order to ensure they have enough testosterone to meet their body’s needs. This won’t be an issue for most men as testosterone is normally a base steroid in a cycle. If it is not used as a base steroid the individual should ensure he administers the minimal amount necessary to combat suppression. Once the cycle of steroids is over, while exogenous testosterone protected the individual while on cycle, at the end of the cycle natural production is still suppressed. Natural production will begin again once all the exogenous hormones have cleared the system, but returning to your prior levels pre-cycle will take a lot of time. In fact, it could potentially take up to a year assuming no other anabolic steroids were used during this period. By implementing a PCT plan, we stimulate natural testosterone production, cut down on the total recovery time and ensure we have enough testosterone for proper bodily functions. This does not bring our total levels back to their previous naturally high state, but it speeds up the recovery and ensures we do not spend a lot of time in a low testosterone state. Not only is a low testosterone condition extremely unhealthy and bothersome due to a host of possible symptoms, it can see the lean tissue gained on cycle destroyed. During a phase of low testosterone, it is easy for cortisol to become dominant in the body, which will destroy muscle tissue and promote fat gain. Due to the need for a strong PCT and Aromasin carrying extremely strong natural testosterone stimulating properties, this makes it very appealing for this purpose. Due to the slight androgenic nature and moderately decent promotion of IGF-1 this makes it even more appealing. However, we must consider the primary purpose of Aromasin, which is as an anti-estrogen. High levels of estrogen can be problematic, but the hormone is still necessary to our body’s health. It is important in maintaining a proper immune system, as well as in the maintenance of healthy cholesterol levels. Then consider the PCT, which in part is primarily designed to stimulate natural testosterone production, but the overall primary point is to normalize the body. We cannot normalize with low estrogen levels. For a proper PCT that not only stimulates testosterone production but promotes overall normalization, SERM’s should always be your first choice. Side Effects of Aromasin: The possible side effects of Aromasin are very similar to the primary AI’s in Arimidex and Letrozole. Many who use the AI often report fatigue and weakness, but this is often not an issue for the anabolic steroid user. The exception would be the steroid user who is in the middle of a harsh cutting cycle, such as in preparation for a bodybuilding contest. Many bodybuilders often report strong lethargy during this period, which isn’t surprising due to the intense diet and often incredible amount of cardio. However, it’s often amplified by the use of an AI like Aromasin. Overall, the primary possible side effects of Aromasin include: Weakness or Fatigue Headaches Hot Flashes High Blood Pressure Joint Pain Depression (rare) Nausea and/or Vomiting (rare) While the above represents the primary possible side effects of Aromasin, studies have shown the AI may have the ability to decrease bone mineral content, which in turn could increase the individual’s risk of osteoporosis. This should not be a large concern for most steroid users as many steroids actually have the ability to greatly increase bone mineral content. Regardless, when looking at the side effects of Aromasin, while they largely revolve around possible the overall chance surrounds the individual’s nature. We all respond to varying medications and hormones differently. This includes AI’s like Aromasin to every last over the counter medication on earth and even applies to many of the foods we eat. The final side effect of Aromasin will revolve around cholesterol. Aromasin, like all AI’s has the ability to negatively skew cholesterol levels. Alone it doesn’t appear to carry this ability at a significant level, but when combined with an aromatizing steroid data shows that it may in fact become significant. This can be an issue of concern for the steroid user as many anabolic steroids already have the ability to negatively affect cholesterol levels. This is an issue that many steroid users give very little attention to. Most are far more concerned with possible visually related side effects such as acne, possible hair loss and water retention, but these really aren’t too concerning. Cholesterol, that is an issue of concern, and while it is very possible for a healthy adult to maintain proper cholesterol levels and use anabolic steroids, it will take some effort and is worthy of your attention. When looking at the hard data at hand, we find that the use of Testosterone at a therapeutic level, such as in the treatment of low testosterone will statistically produce no negative effect on cholesterol levels. However, the same data shows that when the same level of testosterone is conjoined with an AI like Aromasin, HDL cholesterol can be decreased or suppressed by as much as 25%. Then we have performance level doses, which will have a moderate effect on HDL cholesterol, but once again this is exasperated by the use of an AI. Due to the potential negative effect on cholesterol, Aromasin and other AI’s should only be used when necessary. Many anabolic steroid users rely on AI’s heavily and that is a mistake. It is possible to avoid estrogenic side effects without an AI. It’s not always possible, but when possible it should be avoided. Many will find SERM’s like Nolvadex to provide all the protection they need. A SERM will not inhibit aromatization or lower serum estrogen levels, but it will attach to the receptors and prevent estrogen from binding. This can greatly aid in the prevention of gynecomastia. It can help with water retention to a degree, but it’s often not enough for many men. However, most men will find they can do a lot to control water retention if they do a better job controlling their diets. Excess calories are necessary for growth, but when the excess is heavy this will promote water retention. This will hold very true with excess carbohydrates more so than anything else and will hold true with or without the use of anabolic steroids. If the individual is consuming an abundant amount of calories and adds an aromatizing steroid to the mix, this will only exasperate the problem. Further, keep in mind that while excess calories are necessary for growth, normally this only requires a slight increase above maintenance. The total increase will vary from one man to the next based on his need, but rarely is it as abundant as many make it. Control your diet and your carbohydrate intake and you will do a lot for controlling water retention. While SERM’s can offer a lot of protection, some will still need AI’s. This will be very true in many hardcore plans, and can often be beneficial to a contest cycle. However, use should be limited to when only necessary. Many who implement moderate anabolic steroid cycles, which is the vast majority of anabolic steroid users would be surprised by how little Aromasin or any AI they could actually get by with. Aromasin Administration: In a therapeutic setting to treat breast cancer, Aromasin is only used after Nolvadex has failed. This is normally after 2-3 years of Nolvadex therapy. From here Aromasin is given to the patient at a dose of 25mg per day, which will normally last another 2-3 years or until the cancer’s progression has come to a halt. This is normally followed by more Nolvadex therapy in an effort to halt the cancer from returning. This is a highly successful plan in the fight against breast cancer. In a performance setting, standard Aromasin doses will normally be 12.5-25mg every other day. Most should be fine with 12.5mg every other day, with some getting by with only two to three doses per week. The individual’s total sensitivity and the composition of the steroid in cycle in question will dictate the final outcome. There will be, however, some who require a daily dose with as much as 25mg per day. This should be short lived and only continued as long as necessary due to the possible cholesterol issues. This type of use can prove very useful for the competitive bodybuilder 7-14 days leading up to the completion in an effort to come in as dry and hard as possible. But again, this full dose use is only used for a limited time. Availability of Aromasin: Aromasin is widely available on the prescription market and to a degree the black market. Counterfeits do not appear to be a massive problem. However, while some black market suppliers carry it, particularly anabolic steroid suppliers, it is not as common as Arimidex or Letrozole. Regardless of where you find it, the pharmaceutical or black market, the true Exemestane tablet is only found under the Aromasin brand. While the Aromasin tablet is the most common, many research chemical labs (RCL’s) have begun to carry their own Exemestane product. RCL’s are legally allowed to manufacture such products in their liquid state so as long as they are manufactured and sold for research purposes only. While almost all RCL’s carry liquid Anastrozole and Letrozole, some still won’t have liquid Exemestane, but it is rapidly becoming more popular and more and more RCL’s are starting to carry it. Aromasin Reviews: Aromasin is an extremely powerful and valuable AI. We cannot necessarily call it more valuable than the more traditional AI’s, but it is useful. In the end, you may have to try varying AI’s at different times to find which one works best for you. If you are using Aromasin during an anabolic steroid cycle, you are strongly encouraged to keep the possible cholesterol issues in mind. Some have suggested that the use of an AI like Aromasin along with a low dose of Nolvadex could protect the individual from cholesterol issues. While there is no concrete data to fully support this, in theory it may work as Nolvadex as an anti-estrogen actively acts as estrogen in the liver, thereby promoting healthier cholesterol levels. Regardless, for your cholesterol health, ensure your diet and lifestyle is cholesterol friendly. A cholesterol friendly lifestyle will be limited in saturated fats and simple sugars. It should also be abundant in omega fatty acids; daily fish oil supplementation is advised. Incorporating plenty of cardiovascular activity into your routine is also advised. Some may also find a cholesterol antioxidant supplement to be useful.
  3. Anastrozole is an extremely powerful anti-estrogen officially belonging to the Aromatase Inhibitor (AI) family. Developed in the early 1990’s by Zenaca Pharmaceuticals and released in 1995 under the trade name Arimidex, this is perhaps the most commonly used AI and one of the most common anti-estrogens on the market. Arimidex has proven to be very effective in breast cancer treatment, even more so than traditional Nolvadex(Tamoxifen Citrate), and is a favorite anti-estrogen among many anabolic steroid users. Countless anabolic steroid users rely on Arimidex for on cycle estrogenic protection. Many anabolic steroids have the ability to aromatase and lead to excess estrogen, which in turn can lead to some of the most commonly associated side effects of anabolic steroid use. Arimidex Functions & Traits: The functions and traits of Arimidex although powerful are extremely simple. As an AI Arimidex functions by blocking the aromatase enzyme, which is in turn responsible for the production of estrogen. By inhibiting the aromatase process, Arimidex will lower the body’s serum estrogen levels; in fact, a total suppression of estrogen by 80% has been well noted with this AI. This will prove very beneficial to numerous breast cancer patients and extremely valuable to many anabolic steroid users. Arimidex also has the ability to stimulate the release of Luteinizing Hormone (LH) and Follicle Stimulating Hormone (FSH), two hormones essential to natural testosterone production. This has led some physicians to use the AI in low testosterone treatment plans in place of testosterone, but it’s generally not the best choice. Arimidex in a low testosterone plan is generally better served in conjunction with testosterone therapy. We will look more into this when we discuss the effects of Arimidex later on. Effects of Arimidex: As an anti-estrogen, Arimidex is valuable to the breast cancer patient as many forms of breast cancer feed off of the estrogen hormone. While perhaps an oversimplification, by administering Arimidex the effect starves the cancer. For decades Nolvadex was used for this purpose. Nolvadex has the ability to bind to the estrogen receptors, which in turn prevents estrogen from binding. However, AI’s like Arimidex actively inhibit the production of estrogen and reduce the actual amount of circulating hormone. In short, there is no estrogen available to cause damage to the breast cancer patient. In recent years, Arimidex has become the leading anti-estrogen in the treatment of hormone receptor-positive breast cancer, especially among post-menopausal women. Once the cancer has subsided, it is not uncommon for Nolvadex to be introduced in order to keep the cancer at bay. For the anabolic steroid user, the effects of Arimidex are greatly appreciated in its ability to protect against estrogenic related side effects. Many anabolic steroids have the ability to promote estrogenic side effects due to the testosterone hormone’s interaction with the aromatase enzyme. As aromatization occurs, estrogen levels rise and this can lead to gynecomastia and excess water retention. When excess water retention becomes severe, this can also promote high blood pressure. Not all anabolic steroids aromatize, and as such, not all can lead to estrogenic related effects. However, many common steroids do carry the ability to promote estrogenic activity including Dianabol, all forms of Nandrolone and Boldenone to a degree and of course, all forms of testosterone heavily. By including Arimidex in an anabolic steroid cycle that contains aromatizing steroids, the individual can protect against gynecomastia and water retention. This will also protect against high blood pressure. Some steroids can still cause high blood pressure without water retention, but heavy excess water retention is the number one culprit of high blood pressure among anabolic steroid users. Without question, AI’s like Arimidex are the most effective anti-estrogens for combating estrogenic related side effects. SERM’s like Nolvadex can also be useful and while not as effective should be the first choice when possible. Arimidex has the ability to negatively affect cholesterol as we will see in the side effects section. However, we will also find cholesterol issues can be avoided. As a testosterone stimulating compound, Arimidex can be appealing for low testosterone treatment plans and for Post Cycle Therapy (PCT) for anabolic steroid users. In the case of low testosterone treatment, it’s often not enough. However, it can still be beneficial in conjunction with exogenous testosterone therapy in protecting against estrogenic side effects. As for PCT use, some will attempt it and it can have a positive effect, but it is generally not recommended. The main purpose of a PCT plan is to stimulate natural testosterone production in order to protect lean muscle tissue, keep body fat under control and promote a better state of health. However, the overall purpose is normalization, which cannot be reached when using Arimidex post cycle due to the tremendous estrogen reduction. Although high levels of estrogen can be problematic, some is necessary to proper bodily function, especially regarding the immune system and cardiovascular health. For the anabolic steroid user, AI’s should be saved for on cycle use with SERM’s being used for PCT. Side Effects of Arimidex: Arimidex carries with it several possible side effects. Many of the side effects of Arimidex will be response related. Response side effects are common with all medications; some of us can take Aspirin while others can’t. The side effects of Arimidex will also vary depending on anabolic steroid use in a few specific areas. Those who are using Arimidex without anabolic steroids often report weakness and fatigue; in fact, this may be the most common side effect of Arimidex. Most anabolic steroid users will not have this issue with low dose Arimidex use. However, we can make an exception when it is used in hard cutting or competition cycles when calories are very low and training often extremely intense. Other possible side effects of Arimidex use include: Headache Hot Flashes High Blood Pressure Joint Pain Depression (rare) Nausea and or Vomiting (rare) Arimidex studies have also shown that the AI may have the ability to decrease bone mineral content, which in turn could make the individual more susceptible to osteoporosis. This shouldn’t be a big issue for anabolic steroid users as many anabolic steroids have the ability to promote bone mineral content. As for the primary six possible side effects of Arimidex listed above, while possible most adults should be able to use the AI without any related issues, but keep in mind such issues are possible. We all respond to varying medications differently, we even respond to varying foods differently, which can make total response on an individual basis impossible to fully predict. The final issue revolving around the side effects of Arimidex surrounds cholesterol. Arimidex does have the ability to negatively effect cholesterol levels, but alone it doesn’t appear to be significant in most cases. However, when conjoined with anabolic steroid use, specifically an aromatizing steroid like testosterone it appears to be significant. For example, studies have shown that a moderate dose of Testosterone Enanthate for 12 weeks does not appear to have a strong affect on cholesterol. However, when this same dose is coupled with an AI like Arimidex it can suppress HDL cholesterol by as much as 25%. In this case, we’re actually talking about therapeutic level doses as well as performance. True performance doses of testosterone will have a stronger impact on HDL cholesterol, and again around a 20%+ decrease in HDL when conjoined with an AI. Due to the potential cholesterol issues brought on by Arimidex use by the anabolic steroid user, a healthy and cholesterol friendly lifestyle is extremely important. A healthy lifestyle should first and foremost surround your diet. Diets should be low and very limited in saturated fats and simple sugars. They should also be rich in omega fatty acids. Daily fish oil supplementation is advised. It’s also worthwhile to consider the use of a cholesterol antioxidant supplement. And as a final note, if cardiovascular health is to be protected the individual should always incorporate plenty of cardiovascular training into his routine. Daily cardiovascular activity is recommended. Due to the possible cholesterol issues, moderate anabolic steroid cycles may be best served with SERM’s in order to protect against estrogenic related side effects. SERM’s will not negatively affect cholesterol; in fact, SERM’s like Nolvadex have been shown to promote healthy cholesterol levels due to their ability to act as estrogen in the liver. However, for many a SERM won’t be enough and AI’s will be necessary. If an AI is necessary, the individual should limit his use and only use as much as is actually needed. Some have suggested that a 10mg per day dosing of Nolvadex along with your Arimidex use may actually aid in cholesterol management. Arimidex Administration: In the treatment of breast cancer, Arimidex is almost always dosed at 1mg per day until the cancer subsides. Use may continue for a time at this stage and will often be switched to Nolvadex in a preventative measure once the cancer is in remission. For the anabolic steroid user, Arimidex doses can vary with 0.5-1mg every other day being the most common. Very few should ever need more than 1mg every other day and many will be more than fine with half that amount. In therapeutic plans such as low testosterone treatment even less may be needed. We can, however, make an exception in Arimidex doses for competitive bodybuilders. Competitive bodybuilders may find a full 1mg every day the last 10-14 days leading up to competition to be useful. This will greatly aid in hardening, but it will be draining to say the least. Of course, at this stage of a competition diet most have very little energy to begin with anyway. Availability of Arimidex: Arimidex is widely available on the prescription and black markets. In the U.S. it is not classified as a controlled substance, but you will need a prescription to legally obtain it. As for black market purchases, nearly all anabolic steroid suppliers carry Arimidex or another brand of Anastrozole. In recent years, the ability to buy Anastrozole from research chemical labs (RCL’s) has become very popular. RCL’s manufacture various non-controlled substances in their liquid state, often highly concentrated and are able to sell them legally for research purposes only. This is obviously a loophole in the law many anabolic steroid users take advantage of. Regardless of how you obtain it, you will find Arimidex is easier to obtain than many anabolic steroids. Buy Arimidex Online - Warning: Millions buy Arimidex online though anabolic steroid suppliers or RCL’s. The compound is rarely counterfeited; whomever you get it from quality will rarely be an issue. However, if you buy Arimidex online from a steroid supplier you will be breaking the law. Further, while an RCL purchase is legal, it’s only legal for research purposes and this could be made an issue if law enforcement wished to make it one. If you are caught with a supply of anabolic steroids, your “research” claim will be a stretch. In any case, the best way to buy Arimidex will always be through the pharmacy based on the prescription given by your doctor, and it’s not a hard one to get. Due to the laws and varying scenarios that surround compounds like Arimidex and anabolic steroids, you are encouraged to visit the sponsors here at Steroid.com. The sponsors here at Steroid.com can provide you high quality anabolics legally and without a prescription. For those who suffer from low testosterone or think you may suffer from low testosterone, please visit Lowtestosteorne.com. Lowtestosteorne.com can help you with this situation and ensure you legally obtain the testosterone and Arimidex you need to completely remedy your condition. Arimidex Reviews: There are several Aromatase Inhibitors available, Femara (Letrozole), Aromasin (Exemestane) and Arimidex (Anastrozole) being the most common. All three are very similar and while all three carry slight differences that make them unique many agree Arimidex may be the most valuable of all. Arimidex is generally the modern preferred anti-estrogen in breast cancer treatment, as well as the preferred AI in low testosterone treatment plans. For the anabolic steroid user, it is highly efficient and should be the only AI you need. However, in cases where gynecomastia symptoms are already beginning to show, many report heavy Letrozole doses to be the answer to the remedy, where in time switching to Arimidex as a preventative measure. However, in the end, for the performance enhancing athlete, he may need to try all three at varying times to find which AI works best for him.
  4. Superdrol is an anabolic steroid that carries a bit of a unique history compared to many anabolic steroids. Superdrol itself is merely a brand name of an over the counter anabolic steroid sold as a pro hormone or nutritional supplement by Anabolic Extreme. While an anabolic steroid, the active hormone Methyldrostanolone had never been placed on the controlled substance list in the U.S. and in 2005 it would hit the shelves of most major supplement companies and enjoyed massive success. However, in 2006 due to tremendous FDA pressure Superdrol would be discontinued. While the Superdrol brand was short lived, over the counter and black market Methyldrostanolone would continue to appear around the world until mid-2012. In 2012 Methyldrostanolone would be placed on the U.S. controlled substance list and classified as a Schedule III controlled substance along with all anabolic steroids. Methyldrostanolone or Superdrol, while it did not appear on the market until 2005 is not a new anabolic steroid. Syntex first created the Methyldrostanolone hormone in 1959 at the same time as Drostanolone (Masteron) and Oxymetholone (Anadrol). However, the Methyldrostanolone hormone never received a pharmaceutical push like the other two hormones. The exception would be its inclusion in Dimethazine; a compound that metabolically dissolved and converted to Methyldrostanolone post administration. As we dive into the Superdrol compound, as you may have already guessed we will find it is very similar to Drostanolone or the popular anabolic steroid Masteron. Superdrol Functions & Traits: Superdrol is an anabolic androgenic steroid comprised of the active steroidal hormone Methyldrostanolone. This is a dihydrotestosterone (DHT) derived anabolic steroid or more specifically a structurally altered form of Drostanolone. Superdrol is simply the Drostanolone hormone with an added methyl group at the 17th carbon position that allows the hormone to survive oral ingestion and officially classifies it as a C17-alpha alkylated (C17-aa) anabolic steroid. It also carries an added methyl group at the carbon two position, which greatly increases its anabolic power. These slight alterations will also reduce Superdrol’s androgenicity compared to Masteron, which isn’t all that androgenic to begin with. On a structural basis, Superdrol carries an anabolic rating of 400; nearly four times that of Masteron. It will also carry an androgenic rating of 20, which is extremely mild. This is a non-aromatizing anabolic steroid carrying no estrogenic or progesterone activity. When looking at the traits of Superdrol, there is nothing all that remarkable about this steroid compared to many others. The mere fact that it enjoyed years of grey legality is truly the only remarkable attribute. This isn’t to take away from the steroid’s ability, but is merely stated to clear up any confusion or misguided notions. Superdrol will notably enhance protein synthesis and nitrogen retention. Protein synthesis refers to the rate by which cells build proteins and nitrogen represents a key component in muscle tissue composition. The enhancement in both areas promotes a stronger anabolic atmosphere enabling the individual to build more lean tissue or preserve it during a calorie restricted state. The hormone will also significantly increase red blood cell count providing greater muscular endurance. This is due to red blood cells being responsible for carrying oxygen to and through the blood and the increase in cells providing greater blood oxygenation. Effects of Superdrol: When looking at the effects of Superdrol, the best way to describe the steroid as is a total body transforming product. Through its marketing campaign it was touted as being a more powerful mass builder than Anadrol, hence the name Superdrol; a play on words “Super Anadrol.” However, athletes who have used both will attest the effects of Superdrol will in no way lead to mass gains even comparable to Anadrol. However, significant gains in lean tissue can be made so as long as adequate calories are consumed. A gain of 5-10lbs is more than possible and will not be accompanied by the water retention Anadrol often brings. The individual should also find he is able to make cleaner off-season gains due to the effects of Superdrol promoting a stronger metabolism. This is not to say body fat cannot be gained, but you should be able to make better use of your caloric surplus when Superdrol is in play. The effects of Superdrol can also be very beneficial to the dieting athlete as a cutting steroid. This compound will greatly preserve lean tissue during a caloric deficit, a key component to successful dieting. In order to lose body fat we must burn more calories than we consume. This puts lean tissue at risk as the body will take what it needs to meet its energy demands from anywhere it can get it. Due to the body’s natural survival instinct, it will often take energy from muscle tissue rather than body fat. The key to successful dieting is ensuring that not only is fat lost but the lean tissue we hold is preserved. The effects of Superdrol will ensure this goal is met. Through the effects of Superdrol the individual should also notice greatly improved conditioning in terms of a dryer, harder look. This isn’t all that surprising when we consider this steroid is in many ways oral Masteron, a steroid well known for promoting such traits. Regardless of your reason for use, bulking or cutting, the effects of Superdrol will improve recovery and muscular endurance. We cannot call it the strongest steroid in this regard but the improvements will be significant, and as with all steroids the most important. You will not tire out as fast allowing for work to be done at a maximal level for longer periods of time. This does not mean training time frames need to be increased, but rather they become more efficient. The entire point behind anabolic steroid use is to take what you’re already doing right and to simply do it better. Then we have recovery, and this is where the effects of Superdrol as with many anabolic steroids become invaluable. Recovery is where progress is made. Progress isn’t actually made in the gym when training. When training we are actually tearing our muscle tissue down, and when we recover this is where it is built, repaired and becomes stronger. Side Effects of Superdrol: There are possible side effects of Superdrol all users must be aware of. This is not what we’d label an unfriendly anabolic steroid, but the possible side effects of Superdol can be potentially problematic in a few key areas. Those with high cholesterol or existing liver issues must not use this anabolic steroid. If you are healthy enough for use, you will need to put in a good bit of effort into controlling these areas of your health. In order to help you understand the possible side effects of Superdrol, we have broken them down into their separate categories along with all the information you’ll need. Estrogenic: The side effects of Superdrol do not include any of an estrogenic nature. Gynecomastia and water retention will be impossible with this steroid. An anti-estrogen is not necessary due to the use of Methyldrostanolone. Androgenic: The side effects of Superdrol can include those of an androgenic nature. However, due to a low androgenic nature the threshold for such effects should be fairly high with most men. Possible androgenic side effects of Superdrol include acne, hair loss in those predisposed to male pattern baldness and body hair growth. These effects are highly dependent on genetic predispositions, but even if sensitive you will not be able to reduce the androgenicity of this hormone. The Methyldrostanolone hormone is not metabolized by the 5-alpha reductase enzyme making 5-alpha reductase inhibitors like Finasteride useless with this steroid. The androgenic nature of Superdrol can also promote virilization in women. Such side effects of Superdrol include body hair growth, a deepening of the vocal chords and clitoral enlargement. Despite carrying a low androgenic nature the translating androgenic activity in women does appear to be stronger than its rating would imply. Use without virilization is possible, but it will take very low doses. Most women will find other anabolic steroids like Oxandrolone (Anavar) to be better choices. If a female athlete decides to try Superdrol, if virilization symptoms begin to show it should be discontinued immediately. If use is discontinued at the onset of symptoms they will fade away rapidly. If the symptoms are ignored and use continues, they may become irreversible. Cardiovascular: The side effects of Superdrol in this category can be some of the most concerning of all. The Methyldrostanolone hormone can have a strong, negative impact on lipids by significantly lowering HDL cholesterol (good cholesterol) and increasing LDL cholesterol (bad cholesterol). Despite carrying no estrogenic activity, therefore no water retention, Methyltestosterone may also have a negative impact on blood pressure. However, cholesterol issues are far more likely than blood pressure, but both are possible. Due to the possible cardiovascular issues created by Superdrol, a healthy lifestyle will be imperative. Those with high blood pressure or cholesterol should not supplement with this steroid. If you are healthy enough for use a blood pressure and cholesterol friendly lifestyle will be imperative. The individual’s diet should be rich in omega fatty acids; daily fish oil supplementation is highly advised. The individual should also strictly limit saturated fats and simple sugars and ensure he implements daily cardiovascular activity into his routine. The use of a cholesterol antioxidant supplement is also highly advised. Testosterone: The side effects of Superdrol will include natural testosterone suppression in all men who use the steroid, and it will be significant. The use of exogenous testosterone is advised. Those who do not include exogenous testosterone of some form with their Superdrol use will place their body in a low testosterone state. The form of testosterone you choose is inconsequential, all that matters is your body receives the testosterone it needs as this hormone is essential to a healthy a properly functioning body. Once the use of Superdrol has come to an end and all exogenous hormones have cleared the system natural testosterone production will begin again. However, levels will still be low and most are encouraged to implement a Post Cycle Therapy (PCT) program. A PCT program will stimulate natural testosterone production, which will protect your physique as well as your overall health. It will also greatly cut down the total time to recovery. A PCT plan will not return your testosterone levels back to normal on its own, this will take some time, but it will ensure you have enough testosterone for proper bodily function. An important note on natural testosterone recovery – natural testosterone recovery assumes no damage was done to the body due to improper supplementation practices. It also assumes there was no prior existing low testosterone condition. Hepatotoxicity: Superdol, like all C17-aa anabolic steroids, is hepatotoxic and can potentially stress and damage the liver. Use must not be undertaken if the liver isn’t healthy. During use, liver enzyme values will increase in all who use this steroid. However, an increase in liver enzyme values does not equate to damage but is rather an indicator of stress. However, it will lead to damage if possible precautions are not followed. All who supplement with Superdrol must follow the following recommendations: No other C17-aa steroids should be used during Superdrol use. Excess alcohol consumption must be avoided. Heavy alcohol consumption is tremendously stressful to the liver on its own, and with Superdrol use this will lead to severe liver stress and greatly exasperate the probability of liver damage. Most are encouraged to avoid all alcohol consumption during use of this steroid. Keep in mind, the only reason to use this steroid is for performance purposes, and not only will the added alcohol damage your health there is no substance as anti-performance as alcohol. Over the counter medications should be avoided at all times when possible. Many over the counter medications are hepatotoxic, and in many cases, just as if not more than many anabolic steroids. Use should be limited to when only absolutely necessary. Total use should not exceed eight weeks and most will find a total time frame of six weeks to be best. No C17-aa steroids including Superdrol should be used for at least 6-8 weeks post Superdrol use, and a longer time frame of no use will be healthier. The use of a liver detoxification supplement is highly advised when using Superdrol. If you can follow the above guidelines it will be possible to protect your liver’s health, but you will need to keep an eye on it. All who supplement with Superdrol are strongly encouraged to keep a close eye on their blood pressure, cholesterol and liver health. Superdrol Administration: Standard male Superdrol doses will fall in the 10-20mg per day range for 6-8 weeks. This will equate to 1-2 capsules per day taken with food. Those who enjoy a high level of toleration can consider 30mg per day their next go around with the steroid, but this is not advised for most. Doses of 30mg per day or more will greatly stress the liver and caution is strongly advised. Superdrol stacks well with most all anabolic steroid. A simple stack of Superdrol and some form of testosterone is most common and will greatly benefit any bulking or cutting plan. During bulking phases, additional Nandrolone is a very common part of the stack, as is Trenbolone during a cutting phase. There is no reason any man could not enjoy success with such plans. Availability of Superdrol: Due to the compound no longer being sold over the counter the availability of Superdrol is far less than it once was. You will find some Methyldrostanolone compounds on the black market, but even here it’s not what we’d call extremely common. Due to the high availability of other anabolic steroids on the black market there’s never been a strong need for Superdrol or generic versions of this hormone on the black market. Buy Superdrol Online - Warning: You can buy Superdrol online, or rather a Methyldrostanolone hormone. However, it’s not commonly found like Anadrol, Dianabol, or Masteron, but it can be found. You will not, however, find the original Superdrol brand and anyone reporting to sell it is lying to you. If they actually have old bottles of true Superdrol, keep in mind it will have long since expired as it has not been manufactured in several years. Although you may be able to buy Superdrol online, if you do so in the United States you will be breaking the law. In the U.S. anabolic androgenic steroids, now including Superdrol, are classified as Schedule III controlled substances. You must have a prescription in order to legally purchase or possess an anabolic steroid, and Superdrol or Methyldrostanolone is not a steroid you’ll ever receive a prescription for. Those who break the law will be subject to heavy fines and prison when caught. Outside the U.S. you will find steroid laws are commonly far more lenient. You will find some places that are similarly strict, but you will find many where you can buy anabolic steroids over the counter. However, over the counter Methyldrostanolone isn’t common and most countries do not allow online purchasing. Due to the steroid laws of the U.S. and many countries around the world, you are strongly encouraged to visit the sponsors here at Steroid.com. The sponsors here at Steroid.com can provide you with high quality anabolics without a prescription. You can legally purchase these anabolics without a prescription or fear of legal consequence. Superdrol Reviews: Superdrol is a decent anabolic steroid, but we would not call it superior or even “Super” as its marketing campaign once implied. What truly makes this steroid special was a group of men who recognized a hole in the steroid law and were able to capitalize on it, and in turn, make a nice profit. Due to the marketing and ease of purchase that existed for a long time, many athletes fell in love with this steroid, and it is a fine steroid, but there’s nothing magical or superior going on. Superdrol is a very basic anabolic steroid. Superdrol Profile 2a,17a-dimethyl-5a-androst-3-one-17b-o 2a,17a-dimethyl-etiocholan-3-one-17b-ol Molecular Weight: 318 Formula: C21H34O2 Manufacturer: Syntex Effective Dose (Men): 1-2 Tablets/Day Effective Dose (Women): Not Recommended Half-Life: Approx. 8 Hours Detection Time: Unknown Anabolic/Androgenic Ratio: 400/20
  5. Nandrolone Phenylpropionate is an anabolic steroid that is very similar to the popular Nandrolone Decanoate compound. However, Nandrolone Phenylpropionate was the first Nandrolone compound ever commercially sold. Nandrolone Phenylpropionate hit the shelves in the 1950’s and was brought to the market by Organon under the name Durabolin. Soon after Organon would release its Decanoate cousin under the name Deca Durabolin. Nandrolone Phenylpropionate is a small ester base anabolic steroid and is commonly referred to as NPP. This product has never been as popular as the larger ester Decanoate version, in part due to availability; however, in the modern era it has begun to see a resurgence in both use and availability thanks in part due to underground labs. Nandrolone Phenylpropionate carries with it numerous therapeutic and performance benefits. The Nandrolone hormone is the most commonly prescribed anabolic steroid other than testosterone, but the Decanoate version is the most commonly prescribed Nandrolone form. It is one of the most well tolerated steroids in both performance and medical settings, although possible side effects most certainly exist. Nandrolone Phenylpropionate Functions & Traits Nandrolone Phenylpropionate is a 19-nortestosterone (19-nor) anabolic androgenic steroid. The 19-nor classification refers to a structural change of the testosterone hormone in that the carbon atom has been removed at the 19th position. This simple structural change gives us Nandrolone, and by adding the short Phenylpropionate ester we have Nandrolone Phenylpropionate. On the basis of the hormone’s function, Nandrolone Phenylpropionate is identical to Nandrolone Decanoate. Both forms are comprised of the same active hormone. In the case of NPP we have a shorter ester version that gives a larger burst of Nandrolone after injection, but also carries a much shorter half-life. This means Nandrolone Phenylpropionate has to be injected more frequently than its larger ester counterpart if blood levels are to remain stable. Nandrolone Phenylpropionate is slightly more anabolic than testosterone with a rating of 125 compared to testosterone’s rating of 100. It is also significantly less androgenic with a rating of 37 compared to testosterone’s rating of 100. The reduced androgenicity is due to the Nandrolone hormone reducing to dihydronandrolone (DHN) instead of dihydrotestosterone (DHT). This is one of the reasons Nandrolone Phenylpropionate can be well tolerated at higher doses in some men than higher doses of testosterone. Nandrolone Phenylpropionate is also significantly less estrogenic than testosterone. Both Nandrolone and testosterone aromatize, but Nandrolone only does so at approximately 20% the rate of testosterone. Important Note: Nandrolone Phenylpropionate carries a progestin nature, and this will play into the side effects of this hormone. Nandrolone Phenylpropionate carries many positive traits that are similar to many anabolic steroids. However, this compound also carries functional traits that will far outweigh what some steroidal hormones can do. The positive functional traits of Nandrolone Phenylpropionate include: Increased IGF-1 Production: Insulin-Like Growth Factor-1 (IGF-1) is a potent anabolic hormone that is also essential to our body’s ability to recovery. This is a hormone that affects nearly all cells within the human body. Inhibition of Glucocorticoids: Known as stress hormones (cortisol) these hormones are essential to our health and wellbeing. However, glucocorticoids can also promote muscle loss and fat gain when they become dominant. Vigorous activity can lead to increases in stress hormones. Hormones like Nandrolone can reduce the production of stress hormones. Increased Nitrogen Retention: All muscle tissue is comprised of 16% nitrogen. If retention falls we fall into a catabolic state. The more we retain the more anabolic we remain. Increased Protein Synthesis: This refers to the rate in which cells build proteins, the building blocks of muscle tissue. Increased Red Blood Cell Count: Red blood cells carry oxygen to and through the blood. Greater efficiency results in enhanced muscular endurance and recovery. Increased Collagen Synthesis & Bone Mineral Content: This refers to the strength of bones and cartilage and the ability to strengthen and provide healing relief. This will hold true in joints more so than anywhere else. Important Note: It’s often said Nandrolone forces water into the joints, thereby providing relief. This is not physically possible. It is not water, it is the enhancement of collagen synthesis and bone mineral content that provides relief. Nandrolone Phenylpropionate is also well-suited for medical treatment in a host of areas. Although Nandrolone Decanoate is more commonly used, the Phenylpropionate version is still used with some regularity. The use of Nandrolone Phenylpropionate has been proven useful in the treatment of the following: Muscle Wasting Diseases: Cancer, HIV, etc. Improving Geriatric Weakness & Fatigue Anemia Breast Cancer The Treatment of Burn Victims Ulcers Pituitary Dwarfism Development Retardation in Children Osteoporosis Despite a host of benefits and purposes of use, in the U.S. Nandrolone is generally only prescribed for HIV, AIDS and anemia. Its rate of success in other areas is high, but typically use for such areas of medicine is found outside the U.S. Some U.S. physicians have begun to prescribe it for anti-aging purposes, but this still represents a very small fraction of the total prescriptions. Effects of Nandrolone Phenylpropionate Through a thorough understanding of the functions and traits of Nandrolone Phenylpropionate we already have a good understanding of the positive effects of this steroid. However, to put it in terms that a performance athlete can appreciate we can be a little more specific. For the off-season athlete, a bulking cycle, Nandrolone Phenylpropionate is one of the best steroids he can choose to enhance muscularity and size. This is one of the best mass builders available and for many bodybuilders is used in every bulking plan. Despite being a faster acting Nandrolone form growth will not occur rapidly, but it will be steady, even and significant. This is assuming you are eating enough to grow. In order to grow you must consume more calories than you burn. No steroid in the world can change this truth. But you will get more out of your growth with a steroid like Nandrolone Phenylpropionate if you are doing things properly. You should also notice you stay leaner in your off-season due to the significant metabolic effects of the hormone. And when it comes to recovery from strenuous training very few things will beat Nandrolone Phenylpropionate. Nandrolone Phenylpropionate can also be used for cutting cycles, although it’s not commonly thought of as a cutting steroid. This steroid will significantly protect lean muscle mass better than many steroids. When we diet we must burn more calories than we consume. This is the only way body fat can be lost. Unfortunately, this puts lean muscle tissue at risk. When we diet some lean tissue will be lost, but successful dieting limits this loss, and Nandrolone can provide this protective measure. And once again the recovery benefits will be tremendous, especially when recovery can already be incredibly difficult when dieting due to the caloric deficit. The final benefits for performance surround the athlete. Many athletes use low doses of Nandrolone Phenylpropionate for the recovery and joint relief benefits. These are not masking benefits like painkillers provide but true relief. Some may also find strength increases to a degree, although this isn’t a steroid well known for tremendous strength increasing properties. Regardless, this is one of the more common steroids used by athletes. Side Effects of Nandrolone Phenylpropionate There are several possible side effects of Nandrolone Phenylpropionate use, but it is also one of the more side effect friendly. The key to managing and avoiding side effects is understanding how they occur and proper use of the hormone. For most men serious side effects should be completely avoidable. In order to understand the side effects of Nandrolone Phenylpropionate we have broken them down into their individual categories. [1] Estrogenic: Estrogenic side effects of Nandrolone Phenylpropionate are possible. Estrogenic side effects of Nandrolone Phenylpropionate include gynecomastia, water retention and high blood pressure caused by severe water retention. These side effects can be avoided by the use of an Aromatase Inhibitor (AI) such as Anastrozole (Arimidex). The reason for estrogenic side effects is due to the Nandrolone hormone aromatizing. Aromatization refers to the conversion of testosterone to estrogen. However, the rate of aromatization with this hormone isn’t high, but high enough to cause issues in some men. It is also a progestin, and progesterone can activate the mammary tissue and promote gynecomastia in very sensitive men. Estrogenic or progesterone based, AI’s will provide the needed protection. [2] Androgenic: There are possible androgenic side effects of Nandrolone Phenylpropionate, but they are not extremely likely in men. Hair loss in men predisposed to male pattern baldness is possible as is acne in sensitive men. However, when it comes to such effects this is one of the most well tolerated steroids of all. Genetic predispositions will play the largest role. Important Note: The use of a 5-alpha reductase inhibitor will not reduce the androgenicity of Nandrolone; in fact, it will increase it and should be avoided. Although not extremely androgenic the Nandrolone hormone can promote virilization symptoms in women. Virilization symptoms may include body hair growth, a deepening of the vocal chords and clitoral enlargement. Some women can use low doses without issue, but if symptoms occur use should be discontinued immediately. If discontinued at the onset of symptoms they will fade away. If symptoms are ignored and use continues they may become irreversible. [3] Cardiovascular: Nandrolone Phenylpropionate can have a negative impact on HDL cholesterol (good cholesterol) and it can be somewhat more significant than testosterone. This negative effect may be exasperated by the use of an AI. It is more than possible to use Nandrolone Phenylpropionate without cholesterol issues or cardiovascular incident, but a healthy lifestyle is imperative. Regular cardiovascular activity is important as is a cholesterol friendly lifestyle. [4] Testosterone: The use of Nandrolone Phenylpropionate will suppress natural testosterone production. As with all Nandrolone compounds, one injection will suppress nearly if not all your natural testosterone production. Your genetics will not prevent this and it is something that’s completely unavoidable with use. Because of this fact, it is imperative that all men who use this steroid do so in conjunction with some form of exogenous testosterone. This will prevent the individual from falling into a low testosterone condition, which comes with a host of very undesirable symptoms. Once the use of Nandrolone Phenylpropionate has been discontinued and all anabolic steroids have cleared the body, natural testosterone production will begin again. However, it will not occur overnight and will come slowly. Post Cycle Therapy (PCT) is recommended. This will help stimulate the production of natural testosterone and increase the odds of a successful recovery. PCT will not complete recovery, it will still take several months post PCT, but it will give you a better start. Important Note: Natural recovery assumes no damage was done to the Hypothalamic-Pituitary-Testicular-Axis (HPTA) during use and that no prior low testosterone condition existed. [5] Hepatotoxicity: Nandrolone Phenylpropionate is not toxic to the liver. Nandrolone Phenylpropionate Administration In a medical setting standard male Nandrolone Phenylpropionate doses will normally fall in the 50-100mg per week range. For female use, although not commonly prescribed if prescribed it will normally be the 50mg per week range. In almost all medical settings the Decanoate version is what will be prescribed. For the athlete or bodybuilder doses can vary greatly. 100mg per week will provide significant therapeutic advantage with 200mg per week being more common as this will ensure significantly improved recovery. In most performance circles 300-400mg per week will be the common dosing range, and this is a perfect range for building or preserving muscle tissue. Some will use more, but this will increase the risk of side effects. Regardless of the dose use the total dose is normally split into three equal injections per week or planned out on an every other day basis for optimal results. 8-12 weeks is the normal period of use for most athletes. The exception is female athletes who may use the steroid for 4-6 weeks and normally at a dose no more than 50mg per week if virilization is to be avoided. Availability of Nandrolone Phenylpropionate Nandrolone Phenylpropionate is not available on the U.S. pharmaceutical market and is somewhat limited in supply on the world market. It can be found on the black market somewhat commonly, but nowhere near as commonly as Nandrolone Decanoate. Underground labs have started making it with more regularity and it’s not all that difficult to find, but it will normally cost a little more than its larger ester base counterpart. Buy Nandrolone Phenylpropionate - Warning You can buy Nandrolone Phenylpropionate online and for most this is the only way you’ll be able to buy it. However, if you live in the U.S. you will be breaking the law. If you live in the U.S. you must have a prescription. Not only must you have a prescription, but Nandrolone is classified as a Schedule III controlled substance. Those who break the law often find the punishments to be very harsh. The laws are just as strict in many countries but far more lenient in many others. You must know the law as it pertains to where you live before making a purchase. Due to the strict steroid laws in much of the world, if you are looking for quality anabolics we encourage you to visit our site sponsors. Here you’ll find quality products that are legal and do not require a prescription. Nandrolone Phenylpropionate Reviews The Nandrolone hormone is one of the most valuable anabolic steroids of all; top five without a doubt. Medically its an incredible hormone, although the Phenylpropionate version has never been give the full opportunity to shine. This isn’t because of its inferiority, it’s simply that the medical world doesn’t really need more than one Nandrolone hormone and Decanoate is simply the one its chosen. For the steroid user, this steroid can almost be called essential to an off-season mass plan. But when we look at what it can do for recovery and healing it is almost in a class of its own. Couple this with its side effect friendly nature and this steroid is very hard to beat. However, there’s one important thing we’ve yet to address, erectile dysfunction. Nandrolone is well known for causing erectile dysfunction, often referred to as “Deca Dick.” This isn’t the hormone’s fault; it is due to improper use. As a progestin and a hormone that can produce prolactin erection function can be diminished. Keep a balance in your hormone levels and there won’t be an issue
  6. Chemical Composition Chemical Name(s): 17a-methyl-etioallocholan-2-ene-17b-ol 17a-methyl-5a-androst-2-ene-17b-ol Chemical Formula: C20H32O Molecular Weight: 288 Bioavailability: Estimated at 40% Half Life: 9 Hours Average Dose (Stand Alone): 40-60mg/day Average Dose (Stacked): 10-30mg/day Anabolic/Androgenic Ratio: 1200/187 Description Madol a.k.a. desoxymethyltestosterone or DMT, a testosterone derivative and cousin to methyltestosterone has undergone three significant modifications. In short, they include the addition of a methyl group at carbon 17-alpha for safe liver passage, as well as two additional chemical conversions (the addition of a double bond, and the removal of the 3-keto group) which account for both its enhanced anabolic potency and relative bioactivity. Madol has rightfully earned a solid reputation for being an extremely potent muscle and strength gaining oral steroid thats 60% more anabolic (muscle building) than testosterone, yet only 60% as androgenic (impacting male sex characteristics). Steroid Form Madol is often found in 5 and 10 mg tablets. Although no longer available as a prescription drug, Madol is still being produced in underground labs and is readily available on the black market. Since Madol was never officially approved for human use medical prescribing guidelines are not available. However, for athletic purposes the typical effective dosage range is 5-15 mg daily. It should also be noted that like all orals with very short half-lives, the daily dosage should be split in half and taken both early and late (8-12 hours apart in this case) to ensure stable blood serum levels which negate negative side effects. Indications/Purpose & Side Effects For the Indications/Purpose & Side Effects of Madol see the Testosterone Propionate profile. Additional Information Madol produces no aromatization (testosterones conversion to estrogen) which can result in negative estrogen-related side effects. Thus, unlike testosterone, theres virtually zero water retention making it especially ideal for definition purpose. This quality also makes those who administer Madol more resistant to gynecomastia than those who use traditional testosterones. Madol can be effectively used to augment any cycle, and to support sound physiological functions in cycles which contain Winstrol, Primobolan, Deca-Durabolin, Dianabol, Anavar, Oral Turinabol, Equipoise, and Trenbolone. This is one of my personal favorites and very hard to come across. Find a source who has this and you hit the jackpot
  7. Winstrol is a very commonly used anabolic steroid for cutting cycles. While many people will attempt to use Dianabol or even Anadrol for cutting cycles, Ive really never heard of anyone using Stanozolol for anything except a cutting cycle. Its a bit of a one-trick-pony in this respect. Let me repeat that: Stanozolol is a cutting drug. Not many people will argue for its use in a bulking cycle. Its certainly not a very effective compound for treating anemia (1) and thus, one could rightly assume that its role in bulking cycles is very limited. One novel use for Winstrol in any cycle (perhaps even bulking) would be to use it at a very limited dose, in order to lower SHBG. (2) One of the properties of Winstrol is its profound ability to lower SHBG much more than other steroids. A dose of .2mg/kg lowered SHBG significantly, which would in turn, raise the amount of free testosterone circulating in the body. As with 99% of steroids, however, its important to note that suppression of your natural hormonal levels will occur (though perhaps not to the extent that it will with many other steroids).(10) As with running virtually any compound, testosterone supplementation (i.e. running test in a cycle containing Winstrol) is warranted to avoid possible sexual dysfunction. Winstrol & Stanozolol Side Effects Adding it to a heavy bulking cycle could be problematic, as Stanozolol is a 17aa compound, meaning that its been altered to endure the first pass through your liver without being destroyed. This makes it an orally active compound; so many people choose to take the pills which are available from both legitimate pharmaceutical companies as well as Underground Labs. Unfortunately, since it is 17aa, it is also liver toxic& in fact; Stanozolol has one of the worst hepatoxicity (mg for mg) of any steroid. This is the reason its addition to a bulking cycle could be problematic; generally a bulking cycle will be very heavy, dosage wise as well as toxicity-wise. It also has undesirable results on Cholesterol, and a mere 6mgs/day of Stanozolol can lower HDL by 33% and raise LDL by 29% (3). Cardiac Hypertrophy, even at lower doses could be a concern with Winstrol as well (4) Thus, many people limit their intake of Stanozolol to precontest or Summer-cutting types of cycles. Its generally accepted that due to the toxicity issues of Stanozolol, its use should be limited to 6 weeks& as with anything though, many people have run it for up to 12 weeks with no problems. Winstrol & Stanozolol Use Effects I ran Winstrol for about 3 months (12 weeks) at a dose of 100mgs Every Other Day (along with Test prop at 125mgs, every other day) and I suffered no ill-effects. My joints felt fine, and I can say that the only thing which was undesirable about that cycle was the injection pain. Generally, people report a "dry" and less lubricated feeling in their joints when on this drug (fluid retention is nil with Stanozolol), and also a "dry" overall look as regards contest prep. This could be due to a sort of "reverse-osmotic" effect...of course this is speculation, but people do look "dryer" on Winnie, and some even look dryer in the site they inject (more on this later). There are many conflicting reports on tendon strength and Stanozolol, even in medical journals. Some reports state that it weakens tendons, others that it strengthens them (and some speculation on the internet among many "gurus" is that it strengthens them unevenly, leading to possible injury). For this reason, it may be best for athletes in explosive or high-impact sports to stay away from this drug. It has certainly been shown to be beneficial in some bone ailments induced by glucocorticoid induced stress (5) as well as having collagen producing properties (11), but with all of the anecdotal problems athletes have suffered with their joints while on Stanozolol, I simply can not recommend it with confidence to strength/speed athletes. I can say that personally, it was an effective compound for me and did not cause joint duress, but I can do without the discomfort of the shots, and have found other DHT based compounds to be far more effective (Masteron springs to mind). As previously stated, this compound is unique, as it is available in both an oral form as well as an injectable form. Both forms contain the exact same compound, but injecting this compound (and yes, you can drink the injectable version, and no you shouldn't) is superior to ingesting it orally in terms of nitrogen retention (6), and thus one would also imagine, for overall anabolism. Injecting it also has the advantage of avoiding the "first pass" through your liver, and thus places your liver under less stress. Stanozolol (Winstrol) and Women Stanozolol is also one of the few compounds that women can take safely, as its anabolic:androgenic ratio is quite skewed towards anabolism. Its generally accepted that women can tolerate around 5-10mgs a day of this compound. Men, on the other hand can dose themselves in the .5-1.5mg/kg range. I find 100mgs injected every other Day to be sufficient, but of course, even with the injectable form, every day dosing is optimal. I tend to favor DHT based compounds, and have enjoyed great success with a Winstrol/Masteron/Testosterone cycle, but I suspect that replacing the Masteron in that cycle with Trenbolone would prove more beneficial for most bodybuilders seeking to get ripped. Although the anabolic ratio of this product is very high as compared to its androgenic actions, not many people report huge weight gains off of Stanozolol. Also, interestingly, it has a relatively weak AR binding ability (7), which is quite unusual for a "cutting" steroid. Many of the effects of this drug, as relates to building muscle, are probably from its very high protein synthesizing ability (6) (8). In addition, since this compound is derived from DHT, it tends to promote a very nice, "quality" look to the users muscles, with little or no water retention. Winstrol does not aromatize at any rate and has even been speculated to have anti-progestenic properties (in at least some cases, where it may "block" that receptor) (9). If one were to run ancillary compounds with Stanozolol, perhaps Tamoxifen would be appropriate for its beneficial effects on blood lipids, but an anti-estrogen (in its classic sense) would be unwarranted; proper post cycle therapy is still needed, though. Most underground labs produce Winstrol at very reasonable prices, in both an oral as well as injectable form. Unfortunately, production value differs vastly due to the varying size of the Stanozolol powder used to make the injectable version; the finer the powder, the smaller gauge needle it will fit through, and the easier the injection will be. Of course the opposite is also true& In any case, you should be paying under $100 for a 10ml bottle of 100mg/ml concentration, and roughly the same for 100 or so 10mg tablets.
  8. In the eyes of many performance enhancing athletes, the Trenbolone hormone is considered the single greatest anabolic steroid of all time. With Trenbolone, we have one of the most versatile steroids of all time, an anabolic steroid that can be used for nearly any purpose, and moreover at a rate of power that is unmatched. Of course, as you know most Trenbolone comes with the Acetate ester attached, but here we want to talk about Trenbolone Enanthate. Trenbolone Enanthate is the largest ester based version of the hormone; much larger than the Acetate version, and even larger than the once very popular Parabolan (Trenbolone Hexahydrobenzylcarbonate). By its direct mode of action, Trenbolone Enanthate is the same as all other forms; the properties and traits remain the same; however, the large ester attached will affect its mode of action based on time release, duration of activity and even potency will vary. A very powerful steroid indeed, often considered the ultimate steroid for cutting purposes, the Trenbolone hormone is also a fantastic bulking agent and a tremendous strength increasing steroid, but unfortunately Trenbolone Enanthate can be extremely harsh in some individuals. For reasons that may not seem fair, some people will not be able to use Trenbolone Enanthate, and while this is a principle that holds true with all steroids there will be more who cannot touch the Trenbolone hormone than just about any steroid; the majority will be fine, but there will be a larger number that cannot touch it compared to other steroids. With the above in mind, lets take a direct look at Trenbolone Enanthate and the powerful properties it holds. We want to look at its direct mode of action, its traits and benefits as well as possible side effects, and of course, what we can do in-order to prevent them. Well even look at comparisons between this form and other Trenbolone forms, and in doing so determine if Trenbolone Enanthate is for you. Trenbolone Enanthate Nature & Traits: Trenbolone Enanthate is a 19-nortestosterone (19-nor) anabolic androgenic steroid that carries massive anabolic and androgenic ratings of 500 in both categories; this is five times greater than testosterone in both categories. More importantly than the rating, its translating anabolic and androgenic power corresponds perfectly to its ratings; this is important because thats not always the case. For example, steroids like Halotestin and Proviron among others can be misleading based on ratings; Halotestin carries a massive androgenic rating based on its structure but displays no androgenic activity whereas Proviron carries a pretty decent anabolic rating but very low translating anabolic activity; Trenbolone Enanthate translates perfectly. Carrying an active half-life of approximately 8 days, Trenbolone Enanthate carries the longest active half-life of any Trenbolone form; Trenbolone Acetate carries an active half-life of approximately 3 days with Parabolan carrying an active half-life of approximately 6 days. With an 8 day half-life, you could manage with one injection per week; however, in-order to maintain stable levels, an important performance enhancement factor two injections per week or one injection every 4 days will prove to be far more efficient. Carrying a strong progestin nature with absolutely no aromatizing activity, Trenbolone Enanthate carries almost every positive anabolic steroidal trait known to man. While many other steroids carry some of the same properties, Trenbolone Enanthate does so at a rate of power that is second to none. Without question, the most valuable of all these traits is this steroids ability to enhance nutrient efficiency; in short, each and every gram of carbohydrates, fats and proteins you consume becomes more valuable; you utilize each one to a larger degree. For example, and this is probably the best way to look at it, if you have $1 you are able to purchase $1 of goods and services. With the Trenbolone Enanthate steroid present, this is like being able to purchase $10 worth of goods and services with the same $1. This trait is so important, its the very reason the hormonal compound first came to the market; Trenbolone came to the market in the form of Finaplix pellets; small subcutaneous implant pellets used to beef cattle up by increasing their feed efficiency. Beyond nutrient efficiency, Trenbolone Enanthate is one of the best steroids on earth for promoting two of the most common anabolic steroid traits known to man; enhancing protein synthesis and nitrogen retention. Protein synthesis refers to the rate by-which cells build proteins, where nitrogen retention becomes important because the more we retain the more anabolic we remain. All muscle tissue is comprised of approximately 16% nitrogen, and while that may sound like a small amount, if we fall below an optimal state we will enter into a catabolic atmosphere. Its not to hard to see how enhanced nitrogen retention can be beneficial; as for protein synthesis, protein is the building block of muscle, necessary for growth and preservation, once again we have an easy concept to understand. Then we have another big one as Trenbolone Enanthate will increase the release rate of Insulin-Like Growth Factor-1 (IGF-1) better than just about any anabolic steroid on earth. IGF-1 is a potent protein based peptide hormone produced by all human beings that carries tremendous anabolic power and is essential to healing and rejuvenation. So powerful, not only does IGF-1 affect our muscle tissue, but also affects nearly every cell in the body and plays an important role revolving around our ligaments and tendons, central nervous system and even our lungs among other areas. Another common steroidal trait Trenbolone Enanthate carries, although at an unbelievable rate is the increase in red blood cell production. Red blood cells are responsible for carrying oxygen to and through the blood, and the more red blood cells we carry the greater our blood oxygenation levels; this will be extremely important in the benefits section based on muscular endurance. Then theres another common steroidal trait once again at a tremendous rate of power and it surrounds the reduction of glucocorticoid hormones; glucocorticoids are commonly referred to as stress hormones. While necessary to our immune system to a degree, it is very easy for stress, mental and physical to increase these muscle wasting and fat promoting hormones to an unsatisfactory level. When abundant amounts of glucocorticoids are present, especially cortisol, this can make fat loss extremely difficult as well as lean tissue building; in-fact, it can work against you in the opposite fashion. While perhaps a little simplistic, in many ways glucocorticoids are the direct opposite of anabolic androgenic steroids, but thankfully Trenbolone Enanthate can remedy this problem. As you can see, Trenbolone Enanthate carries numerous traits, but were not done yet. As is with most anabolic steroids, Trenbolone Enanthate will enhance your overall metabolic rate; however, it will go a step further. This is a steroid that binds firmly to the androgen receptor, and as a result directly promotes lipolysis; thats correct, Trenbolone Enanthate will directly promote fat loss. While its not the only steroid that carries this trait, when it comes to a fat burning steroid the Trenbolone hormone is king. The Benefits of Trenbolone Enanthate: In the eyes of many, the Trenbolone hormone is considered the ultimate in cutting cycles; thats not surprising with its strong metabolic increasing and fat burning properties. While those are tremendous benefits, where Trenbolone Enanthate truly shines is in its ability to greatly preserve lean muscle tissue; perhaps better than any anabolic steroid on earth. When we diet, in-order to lose body fat, not weight but body fat we must be in a caloric deficit; we must burn more calories than we consume. As a result, as the body fights change with a desire to hang onto stored body fat due to its survival nature lean muscle tissue is often sacrificed in-order to meet its energy needs. As we lose more lean muscle tissue, this slows down the metabolic rate, and of course, it makes the physique look worse; Trenbolone Enanthate will prevent this. Of course, it gets even better; through its traits, Trenbolone Enanthate will provide the ultimate in visual conditioning effects; were talking about the promotion of a dry, hard physique, and no steroid does it better. Beyond cutting, the benefits of Trenbolone Enanthate are tremendous when it comes to off-season bulking plans; with nutrient efficiency being promoted to such a strong degree along with all its other anabolic promoting effects this isnt hard to see. It is true, Trenbolone Enanthate is not going to pile weight on your frame at the rate of Anadrol or Dianabol; however, this non-aromatizing steroid will pile on nothing but lean tissue with no water weight due to its use, and with adequate calories it will be a significant gain. Further, and this is the big one, due to its metabolic increasing nature, Trenbolone Enanthate will enable you to gain more lean mass with less body fat accumulation that often accompanies off-season bulking phases, and this is invaluable. In-order to gain new lean tissue, unlike dieting you must be in a caloric surplus; your daily caloric intake must be slightly above maintenance. Of course, this will promote fat gain as well; however, Trenbolone Enanthate will minimize it. When it comes to the benefits of Trenbolone Enanthate, we could easily end our discussion with the above and youd already have a fantastic anabolic steroid, but Trenbolone continues to not disappoint. This is a steroid that will greatly increase muscular endurance, more work can be done and you will not tire out as fast. Of course, it will also play an important role in recovery and healing, but there is an interesting note. Some studies have shown the raw power of Trenbolone to be so great and extreme this enhanced rate actually weakens the tendons; however, more studies have shown the opposite affect; real life evidence shows only the positive. It should also be noted; some may find cardiovascular endurance to be slightly decreased with this steroids presence; however, it appears to be a little hit or miss meaning it doesnt appear to affect everyone in this way. The Side Effects of Trenbolone Enanthate: Theres no way to deny it; when it comes to the side effects of Trenbolone Enanthate we have one of the potentially harshest steroids on earth. As well see, this is a steroid that carries many traditional possible anabolic steroid side effects; however, it carries a group that is largely unique unto its own, and unfortunately that is very difficult to predict. As a non-aromatizing steroid, and as a result one that carries no testosterone to estrogen conversion many assume gynecomastia is of no concern; they would be wrong. As a 19-nor anabolic steroid, Trenbolone Enanthate carries a strong progestin nature, and progesterone can induce gynecomastia; however, it is typically only a problem in men who are sensitive to the condition. While a non-aromatizing steroid, Aromatase Inhibitors will protect against progesterone induced gynecomastia, and as youll more than likely be supplementing with testosterone too an Aromatase Inhibitor is a pretty good idea. This leads to another important point; Trenbolone Enanthate, as with all Trenbolone and 19-nor anabolic steroids is as suppressive to natural testosterone as a steroid can be. For this reason, exogenous testosterone supplementation is necessary in-order to prevent not only a potentially bothersome but extremely unhealthy low testosterone condition. The form of testosterone you choose does not matter; all that matters is you provide enough testosterone for your body for proper and healthy function. Beyond gynecomastia, Trenbolone Enanthate can promote high blood pressure; however, this one appears to be largely dose dependent. If you already suffer from high blood pressure, you should not touch this or any anabolic steroid, but if youre healthy and supplement with responsible doses and continue to live in a way that promotes the continuation of healthy levels you should be fine. The same can be said of cholesterol; however, to a lesser degree. Despite lacking no direct dihydrotestosterone (DHT) nature, Trenbolone Enanthate can be very unfriendly to the scalp; men who are predisposed to male pattern baldness will more than likely lose some of their hair; men who are not predisposed have no concern. Further, due to its extreme androgenic activity, the Trenbolone hormone can have a negative impact on the prostate by way of causing prostate enlargement; however, it can be dose dependent as well as surround other anabolic steroids being used such as those with a strong DHT nature. At any rate, it is imperative you do not supplement if you already suffer from prostate issues, and just as important you supplement with responsible doses for responsible periods of time; you must not supplement with the Trenbolone hormone indefinitely or you will greatly risk damage to your prostate. It should also be noted; the Trenbolone hormone appears to be one of the few anabolic steroids that do not carry the C17-alpha alkylated (C17-aa) nature that can increase liver enzymes, and as a result it should be treated as if it were a C17-aa anabolic steroid. Further, in some men it can cause undue stress to the kidneys; use must be of a responsible nature or you can easily get into trouble. The above largely represents the side effects of Trenbolone Enanthate most will need to concern themselves with; however, as mentioned there is a grouping that is a bit unique to this compound. There are four specific side effects of Trenbolone Enanthate that while they can be dose dependent they are in most cases dependent on your individualistic nature; in short, your personal response. In some ways, these side effects will not seem like much, they include anxiety, insomnia, night sweats and rapid heart rate. Such effects can be so harsh, they will display themselves in ways you cannot imagine, and far beyond what any man can tolerate. If such effects occur, you can try lowering your dose, but more than likely youll need to discontinue supplementation altogether. If your dose is of a responsible nature and such effects occur, unfortunately, this probably means the Trenbolone hormone is not for you. It may not seem fair, and maybe its not, but thats life; its not always fair. Comparing Trenbolones: With many Trenbolone forms available, three common forms, a common question is which form of Trenbolone should you choose? Of the three common forms, Trenbolone Acetate is the most powerful on a per milligram basis as its ester takes up less mass in the compound than any other form; more of the mass is actual Trenbolone. Further, it is much easier to maintain stable and peaked blood levels with the Acetate form, and this raises a question; why would we ever consider Trenbolone Enanthate? The only reason you might choose Trenbolone Enanthate over the often viewed superior Acetate version is based on injection frequency; Trenbolone Enanthate only has to be injected twice a week or once every four days, whereas the Acetate version must be injected every other day. Even so, while this is the largest difference, many report the benefits of the Acetate version are more effective and efficient than the Enanthate version; you may have to find out for yourself. It should be noted; theres really no distinct benefit when it comes to Parabolan; however, its the most expensive due to myths and legends that surround it, and one of the most expensive steroids out there in many cases. When deciding on a Trenbolone form, there is an important note; if you have never supplemented with Trenbolone before your first time must not be with Trenbolone Enanthate. If you end up being a poor responder and you have Trenbolone Enanthate in your system, even after you discontinue use you will have to wait weeks before the side effects dissipate due to the large ester. If its your first time, only choose the Acetate version, and if you run into trouble you can discontinue and the side effects will fade away in a few days. If you supplement with the Acetate version and enjoy a positive response, your next go around and then and only then can you consider Trenbolone Enanthate
  9. Oral Turinabol was first developed by scientists in East Germany for their Olympic and national-level athletes to use. This, plus the eventual removal of it from the market caused Oral Turinabol to become a very "sexy" drug for athletes to try and obtain. The East Germans studied this drug pretty extensively for many years and some of the success of this now defunct country was attributed to this drug, which made its first appearance to athletes in East Germany as little blue "Vitamins" their coaches gave to them. This drug has been discontinued by all of the major pharmaceutical houses, and is only found through certain underground labs. Even though some UnderGround Labs have access to this item, and it appears on their price-lists, its still rare enough. I believe it was first produced in the last half decade by a certain cat in Thailand. Its my speculation that its on the cusp of either becoming very popular, to the point where every Underground Lab will start carrying their own version of it, or it will disappear again and only be carried by a select few, if any, suppliers. he easiest way to explain this drug is that it is a derivative of Dianabol. Though it is a derivative of our old friend Diana, its still quite different...remember, Equipoise is estrified Dianabol, and really has nothing in common with it, in terms of real-world-effects. Lets examine Oral Turinabol in relation to D-bol for now, though. The first similarity between the two is that they have both been 17-alpha-alkylated (a carbon atom was added at the 17th position) to survive the first pass through the liver. This, of course, increases hepatoxicity (liver toxicity). Oral Turinabol has a much lower level of androgenic activity compared to dianabol, but a better balance/ratio of anabolic and androgenic effects. It has a rating of a 0 (according to the Vida reference) for androgenic properties and a 53 for anabolic properties based on a score of 100 each for testosterone. This promotes more of a "hard" look, of what competition bodybuilders often call "quality" muscle. You do not get the same "puffy" look as you would on d-bol, and many people have thus compared the results theyve gotten from Oral Turinabol to Anavar. Actually, though, this stuff is simply dianabol with a 4-chloro alteration, the same alteration found in Clostebol. Due to this 4-chloro substitution in the A-Ring of its Steran Nucleus, this drug cannot be aromatized (3). This is, as you know, quite beneficial and is one of the reasons Oral Turinabol has been called a "gentle d-bol." You will probably not get any typical estrogenic side effects like water retention, acne, gyno, etc, at any dose of this drug. A couple of studies I read examining male athletes over a period of six weeks were given 10 mg Oral Turinabol/day did not show any indications of health-threatening effects. It has been recommended that men should take between 20-40mg every day and women a 5mg every day, and I generally think that it is not very strong (as compared to many other orals) and wouldnt drop below the 40mg mark if I were to use it personally. It may perhaps be used in low(er) doses if it is simply being used for its ability to reduce SHBGs binding (1) to other steroids. In this respect, it may have synergy with other drugs, since it has the ability to reduce SHBG and thus free up more testosterone for use in your body. The only negative thing I have heard about this drug is that in high doses (10+mg) virilization has been seen in women(14) and there has been at least one case of testicular tumors, and one case of a guy who suffered adverse effects from 5 years of high-dose use of Oral Turinabol (2)(4). It should be noted that the former East Germans did many experiments with this drug in high doses though, and found it to be a very suitable compound for their athletes. Many of the women suffered virilization at higher doses, though. During the 68-72 Olympic cycles, the East German Sports Oral Turinabol program made its biggest impact. It was around this time, that the East German weightlifters were taking over 10g/year of Oral Turinabol, and their leading male sprinter was taking under 730mgs/year of Oral Turinabol (14). I think this tells me that for real weight gains, and huge gains in the weight room, youre going to need bank-breaking dosages of this stuff. On the bright side, if you are an athlete looking to get faster, a little bit of Oral Turinabol will get you there pretty easily, and with minimal (if any) side effects). I think that its inability to cause negative side effects, and its ability to produce a favorable increase in lean body mass and thus a favorable increase in strength/speed and an athletes strength:bodyweight ratio is what turned the East German coaches and scientists on. It must be noted that, at the time, this stuff was mostly undetectable, and that was certainly a sought after trait by the East Germans, who were looking to circumvent the drug testing procedures of the IOC. Now, of course, Oral Turinabol is detectable, as once its administered to man, three major metabolites are formed: 6 beta-hydroxy-turinabol, 6 beta, 12-dihydroxy-turinabol, and 6 beta, 16-dihydroxy-turinabol (5)(8)(9).All of those metabolites are now detectable by drug screeners. In much smaller quantities at least another three metabolites are excreted, one of which could be identified as 17 epi-turinabol (5), and is easily detected by modern drug tests... No measurable amounts of Oral Turinabol itself is detected in any of the urine samples investigated in sports doping procedures, but the presence of the metabolites is enough to warrant a positive result, and a failed test. Keeping all of this in mind, it is still important to note that the rate of metabolism and urinary excretion or Oral Turinabol is reasonably fast (5), even though it is technically eliminated biphastically (in two stages) by the body, with a terminal 16hr life (1). I think that the sports-doping-party-poopers (The NCAA and IOC) Oral Turinabol is notorious for increasing the time it will take for your blood to clot because it has spontaneous fibrinolytic properties. "Fibrinolytic effects" means that the destruction of fibrin (an insoluble fibrous protein produced in the liver from the soluble protein) is happening in your body. Fibrinogen is important during the blood clotting process, as it is a soluble protein in the blood that is converted to insoluble fibrin by the action of the enzyme thrombin in response to tissue damage. (6)(7) Thus, you will bleed for longer than usual when on this stuff, combine that with the fact that steroids raise your hematocrit and youll be spending your entire morning trying to stop the bleeding if you cut yourself shaving. Well, thats probably an exaggeration, but not by much.
  10. Testosterone Propionate is the shortest-estered testosterone product available. There are some advantages and disadvantages to this. The major disadvantage is that users will have to inject Test Prop at least every other day throughout its cycle to get proper results. The advantages, however, are less bloating and water retention that longer-estered products and because there is less ester in each vial, there is more actual testosterone per injection, which brings better results. Testosterone is the male sex hormone responsible for many of the physical and emotional traits of men. It creates the deeper voices, sex drive, aggression and, of coarse, larger muscles in men. Testosterone makes the muscles retain more nitrogen, which in turn makes the muscle synthesize proteins better, producing larger muscles. The downside to testosterone steroids is that they aromatize, or turn into estrogen, in the body. When the body has too much estrogen it begins to take on female characteristics gynocomastia, water retention, fat gain, loss of sex drive and testicular shrinkage are all most certain side effects of taking testosterone and letting it aromatize in the body. Testosterone propionate is a commonly manufactured, oil-based injectable testosterone compound. The propionate ester will slow the rate in which the steroid is released from the injection site, but only for a few days. Testosterone propionate is therefore much faster acting than other testosterone esters such as cypionate or enanthate, and requires a much more frequent dosing schedule, in order to maintain stable blood levels. While cypionate and enanthate are injected on a weekly or bi-weekly basis, propionate is usually injected every second. The propionate ester can be very irritating to the site of injection. In fact, many sensitive individuals choose to stay away from this steroid completely, their body reacting with a pronounced soreness and low-grade fever that may last for a few days. Those who do not mind frequent injections will find propionate to be quite an effective steroid. As with all testosterones, it is a powerful mass drug, capable of producing rapid gains in size and strength. At the same time the buildup of estrogen and DHT (dihydrotestosterone) will be pronounced, so typical testosterone side effects are to be expected. Many consider propionate to be the mildest testosterone ester, and the preferred form for the dieting/cutting phases of training. Some will go so far as to say that propionate will harden the physique, while giving the user less water and fat retention than one typically expects to see with a testosterone. Realistically however, this is nonsense. The ester is removed before testosterone is active in the body, and likewise the ester cannot alter the activity of the parent steroid in any way, only slow its release. We can say that propionate might be the favored testosterone among female bodybuilders (for those who insist on testosterone use), as blood levels are easier to control with it compared to other esters. Should virilization symptoms develop, one would not wish to wait the weeks needed for testosterone concentrations to fall after a shot of enanthate for example. During a typical cycle one will see action that is consistent with a testosterone. Users sensitive to gynecomastia and water retention may therefore need to add an anti-estrogen like Arimidex, Femara or Aromasin. Those particularly troubled by gynecomastia may find that a combination of Nolvadex and Proviron works especially well at preventing/halting this occurrence. Also unavoidable with a testosterone are androgenic side effects like oily skin, acne, increased aggression and body/facial hair growth. Those who may have a predisposition for male pattern baldness may also find that propionate will aggravate this condition. To help combat this one may choose to Propecia/Proscar, which will reduce the buildup of DHT in many androgen target tissues. This will help minimize related side effects (particularly hair loss) although it offers us no guarantees. And as with all testosterone products, propionate will also suppress endogenous testosterone production. The use of a testosterone stimulating drug like HCG and/or Clomid/Nolvadex is therefore a requirement in order to avoid enduring a post-cycle crash. The most common dosage schedule for this compound (men) is to inject 50 to 100mg, every day or 2nd day. As with the more popular esters, the total weekly dosage would be in the range of 300-700mg. As with all testosterone compounds, this drug is most appropriately suited for bulking phases of training. Here it is most often combined with other strong agents such as Dianabol, Anadrol, or Deca-Durabolin, combinations that prove to work quite well. Propionate however is sometimes also used with nonaromatizing anabolics/androgens during cutting or dieting phases of training, a time when it’s fast action and androgenic nature are also appreciated. Popular stacks include a moderate dosage of propionate with an oral anabolic like Winstrol (15-35 mg daily), Primobolan (50-150mg daily) or oxandrolone (15-30mg daily). Provided the body fat percentage is sufficiently low, the look of dense muscularity can be notably improved (barring any excess estrogen buildup from the testosterone). One could also add a non-aromatizing androgen like trenbolone or Halotestin, which should have an even more extreme effect on subcutaneous body fat and muscle hardness. Of course with the added androgen content any related side effects will become much more pronounced. Women who absolutely must use an injectable testosterone should only use this preparation. The dosage schedule should also be more spread out for a female bodybuilder, with injections coming every 5 to 7 days. The dosage obviously would be lower as well, generally in the range of 25mg to 50mg per injection. Androgenic activity should be less pronounced with this schedule, giving blood levels time to sufficiently decrease before the drug is administered again. In order to further reduce any risks, the duration of this cycle should not exceed 8 weeks. Should a stronger anabolic effect be needed, a small amount of Durabolin (Deca-Durabolin if unavailable), Oxandrolone or Winstrol could be added. Of course the risk of noticing virilizing effects from these drugs may increase, even with the addition of a mild anabolic. Since many of the masculinizing side effects of steroid use can be irreversible, it is very important for the female athlete to monitor the dosage, duration and incidence of side effects very closely. Some Vet companies as well as UG labs are now even producing 250mg/ml dosage vials. This dosage is more shocking than it sounds at first next to all the 250mg enanthate and now cypionate products in circulation. Testosterone propionate is less oil soluble than Testosterone enanthate or cypionate, making a high dosage more difficult to achieve. Before this the highest concentration you could find of this steroid was 100mg/ml. Reaching 250 milligrams is no doubt a result of not simply adding more steroid to one ml of oil, but increasing the alcohol content in the solution considerably as well. This makes for a much more uncomfortable solution to inject. Although admittedly the highest dose of propionate you will ever find, users have been reporting that it is also intolerably painful. Most find they have to dilute the solution with other lower dosed steroids if they are to continue using the product. This should be no a surprise I guess with a steroid that already has a reputation as being painful to inject.
  11. Testolent is the name given to testosterone with the phenylproprionate ester. This particular ester is a medium length ester that falls squarely between testosterones long ester (cypionate) and short ester (propionate). Injections of twp to three times per week are appropriate for this steroid. As with any testosterone, Testolent will give the user more mass to the muscle, burn fat in the body, enhance libido, increase immunity and increase energy. All the usual side effects of testosterone can also be expected conversion to estrogen and DHT, gynocomastia and water-retention.
  12. Testosterone enanthate Testosterone heptanoate; 17b-Hydroxyandrost-4-en-3-one-17-ethanate Molecular Formula C26H40O3 Molecular Weight 400.60 CAS Registry Number 315-37-7 EINECS 206-253-5 Melting point 34-39 ºC alpha 77 º Test Enanthare is one of the most popular used testosterone products on the market today. It is very effective in building muscle, burning fat and gaining strength. It is also cheap and easy to obtain. Testosterone is the male sex hormone responsible for many of the physical and emotional traits of men. It creates the deeper voices, sex drive, aggression and, of coarse, larger muscles in men. Testosterone makes the muscles retain more nitrogen, which in turn makes the muscle synthesize proteins better, producing larger muscles. The downside to testosterone steroids is that they aromatize, or turn into estrogen, in the body. When the body has too much estrogen it begins to take on female characteristics gynocomastia, water retention, fat gain, loss of sex drive and testicular shrinkage are all most certain side effects of taking testosterone and letting it aromatize in the body. Testosterone enanthate is an oil based injectable steroid, designed to slowly release testosterone from the injection site (depot). Once administered, serum concentrations of this hormone will rise for several days, and remain markedly elevated for approximately two weeks. It may actually take three weeks for the action of this drug to fully diminish. For medical purposes this is the most widely prescribed testosterone, used regularly to treat cases of hypogonadism and other disorders related to androgen deficiency. Since patients generally do not selfadminister such injections, a long acting steroid like this is a very welcome item. Therapy is clearly more comfortable in comparison to an ester like propionate, which requires a much more frequent dosage schedule. Testosterone is a powerful hormone with notably prominent side effects. Much of which stem from the fact that testosterone exhibits a high tendency to convert into estrogen. Related side effects may therefore become a problem during a cycle. For starters, water retention can become quite noticeable. This can produce a clear loss of muscle definition, as subcutaneous fluids begin to build. The storage of excess body fat may further reduce the visibility of muscle features, another common problem with aromatizing steroids. The excess estrogen level during/after your cycle also has the potential to lead up to gynecomastia. Adding an ancillary drug like Nolvadex and/or Proviron is therefore advisable to those with a known sensitivity to this side effect. The anti-aromatase Arimidex, Femara, or Aromasin are a much better choices though. It is believed that the use of an anti-estrogen can slightly lower the anabolic effect of most androgen cycles (estrogen and water weight are often thought to facilitate strength and muscle gain), so one might want to see if such drugs are actually necessary before committing to use. A little puffiness under the nipple is a sign that gynecomastia is developing. If this is left to further develop into pronounced swelling, soreness and the growth of small lumps under the nipples, some form of action should be taken immediately to treat it (obviously quitting the drug or adding ancillaries like Nolvadex). Being a testosterone product, all the standard androgenic side effects are also to be expected. Oily skin, acne, aggressiveness, facial/body hair growth and male pattern baldness are all possible. Older or more sensitive individuals might therefore choose to avoid testosterone products, and look toward milder anabolics like DecaDurabolin or Equipoise which produce fewer side effects. Others may opt to add the drug Proscar/Propecia, which will minimize the conversion of testosterone into DHT (dihydrotestosterone). With blood levels of this metabolite notably reduced, the impact of related side effects should also be reduced. With strong bulking drugs however, the user will generally expect to incur strong side effects and will often just tolerate them. Most athletes really do not find the testosterones all that uncomfortable (especially in the face of the end result), as can be seen with the great popularity of such compounds. Although this particular ester is active for a much longer duration, most prefer to inject it on a weekly or bi-weekly basis in order to keep blood levels stable. The usual dosage would be in the range of 250mg-750mg a week. This level is quite sufficient, and should provide the user a rapid gain of strength and body weight. Above this level estrogenic side effects will no doubt become much more pronounced, possibly outweighing any new muscle gained. Those looking for greater bulk would be better served by adding an oral like Anadrol or Dianabol, combinations which prove to work great. If one wishes to use a testosterone yet retain a level of quality and definition to the physique, an injectable anabolic like DecaDurabolin or Equipoise may prove to be a better choice. Here we can use a lower dosage of enanthate, so as to gain an acceptable amount of muscle but keep the buildup of estrogen to a minimum. With the proper administration of ancillary drugs, Nolva/Clomid and HCG, during post cycle recovery, much of the new muscle mass can be retained for a long time after the cycle has been stopped.
  13. Testosterone Cypionate is the longest-estered testosterone available today. It has a half-life in the body of 15 to 16 days and is found as injectable oil. Because it reacts in the body for so long, it can cause more water retention than other steroids and is best used as bulking compound in a stack. Testosterone is the male sex hormone responsible for many of the physical and emotional traits of men. It creates the deeper voices, sex drive, aggression and, of coarse, larger muscles in men. Testosterone makes the muscles retain more nitrogen, which in turn makes the muscle synthesize proteins better, producing larger muscles. The downside to testosterone steroids is that they aromatize, or turn into estrogen, in the body. When the body has too much estrogen it begins to take on female characteristics gynocomastia, water retention, fat gain, loss of sex drive and testicular shrinkage are all most certain side effects of taking testosterone and letting it aromatize in the body. American athletes have a long and fond relationship with Testosterone cypionate. While Testosterone enanthate is manufactured widely throughout the world, cypionate seems to be almost exclusively an American item. It is therefore not surprising that American athletes particularly favor this testosterone ester. But many claim this is not just a matter of simple pride, often swearing cypionate to be a superior product, providing a bit more of a “kick” than enanthate. At the same time it is said to produce a slightly higher level of water retention, but not enough for it to be easily discerned. Of course when we look at the situation objectively, we see these two steroids are really interchangeable, and cypionate is not at all superior. Both are long acting oil-based injectables, which will keep testosterone levels sufficiently elevated for approximately two weeks. Enanthate may be slightly better in terms of testosterone release, as this ester is one carbon atom lighter than cypionate (remember the ester is calculated in the steroids total milligram weight). The difference is so insignificant however that no one can rightly claim it to be noticeable (we are maybe talking a few milligrams per shot). Regardless, cypionate came to be the most popular testosterone ester on the U.S. black market for a very long time As with all testosterone injectables, one can expect a considerable gain in muscle mass and strength during a cycle. Since testosterone readliy converts to estrogen, the mass gained from this drug is likely to be accompanied by quite a bit of water retention. The resulting loss of definition of course makes cypionate a very poor choice for dieting or cutting phases. The excess level of estrogen brought about by this drug can also cause one to develop gynecomastia rather quickly. Should one notice an uncomfortable soreness, swelling or lump under the nipple, an ancillary drug like Nolvadex should be added immediately. This will minimize the effect of estrogen greatly, making the steroid much more tolerable to use. The powerful anti-aromatases Arimidex, Femara, or Aromasin are yet a better choice. Those who have a known sensitivity to estrogen may find it more beneficial to use ancillary drugs like Nolvadex and Proviron from the onset of the cycle, in order to prevent estrogen related side effects before they become apparent. Since testosterone is the primary male androgen, we should also expect to see pronounced androgenic side effects with this drug. Much intensity is related to the rate in which the body converts testosterone into dihydrotestosterone (DHT). This, as you know, is the devious metabolite responsible for the high prominence of androgenic side effects associated with testosterone use. This includes the development of oily skin, acne, body/facial hair growth and male pattern balding. Those worried that they may have a genetic predisposition toward male pattern baldness may wish to avoid testosterone altogether. Others opt to add the ancillary drug Proscar/Propecia, that prevents the conversion of testosterone to dihydrotestosterone. This can greatly reduce the chance for running into a hair loss problem, and will probably lower the intensity of other androgenic side effects. Although active in the body for much longer time, cypionate is injected on a weekly or bi-weekly basis in order to maintain stable blood levels. At a dosage of 250mg to 800mg per week we should certainly see dramatic results. It is interesting to note that while a large number of other steroidal compounds have been made available since testosterone injectables, they are still considered to be the dominant bulking agents among bodybuilders. There is little argument that these are among the most powerful mass drugs. When taking dosages above 800-1000mg per week there is little doubt that water retention will come to be the primary gain, far outweighing the new mass accumulation. The practice of “megadosing” is therefore inefficient, especially when we take into account the typical high cost of steroids today. It is also important to remember that the use of an injectable testosterone will quickly suppress endogenous testosterone production. It is therefore mandatory to complete a proper post cycle therapy, constisting of HCG and Clomid or Nolvadex at the conclusion of a cycle. This should help the user avoid a strong “crash” due to hormonal imbalance, which can strip away much of the new muscle mass and strength. This is no doubt the reason why many athletes claim to be very disappointed with the final result of steroid use, as there is often only a slight permanent gain if anabolics are discontinued incorrectly. Of course we cannot expect to retain every pound of new bodyweight after a cycle. This is especially true whenever we are withdrawing a strong (aromatizing) androgen like testosterone, as a considerable drop in weight (and strength) is to be expected as retained water is excreted. This should not be of much concern; instead the user should focus on ancillary drug therapy so as to preserve the solid mass underneath. Another way athletes have found to lessen the “crash”, is to first replace the testosterone with a milder anabolic like Deca-Durabolin. This steroid is administered alone, at a typical dosage (200-400mg per week), for the following month or two. In this “stepping down” procedure the user is attempting to turn the watery bulk of a strong testosterone into the more solid muscularity we see with nandrolone preparations. In many instances this practice proves to be very effective. Of course we must remember to still administer ancillary drugs at the conclusion, as endogenous testosterone production will not be rebounding during the Deca therapy.
  14. Understanding Testosterone-Suspension As by its nature Testosterone-Suspension functions by the same mode of action as all testosterone compounds. As Suspension, as it is commonly referred has no ester attached the entire mass of the compound is pure testosterone. For example, Testosterone-Propionate, because part of the compounds mass is the Propionate ester, 100mg will yield approximately 83mg of testosterone; conversely, because there is no ester in the Suspension form 100mg of Testosterone-Suspension will yield exactly 100mg of active testosterone. As there is no ester attached the compound becomes active almost immediately once injected; however, because there is no ester attached testosterone levels fall dramatically and rapidly; one injection of Testosterone-Suspension, assuming no other testosterone is administered will be used in in approximately one day. For this reason, when it is used necessarily daily injections will prove to be the only method of application. The Functions of Testosterone-Suspension As Testosterone-Suspension is simply testosterone, the benefits provided via its function are the same as all forms of testosterone and to understand them we only need to understand the active hormone itself. Testosterone is a hormone produced naturally by the body imperative for a host of functions. When testosterone levels become low we suffer, we they are adequate we thrive and when testosterone levels exceed natural production we enhance the functions it naturally provides. As by its mode of action Testosterone-Suspension greatly increases nitrogen retention in the muscles allowing for increased protein absorption and storage; as protein is a key in growth and preservation this is an invaluable trait. Further, Testosterone-Suspension dramatically increases red blood cell mass and counts aiding in performance and creating a playing field apt for an anabolic nature. As Testosterone-Suspension is both highly anabolic and androgenic, equal on both counts, by the environment it creates it provides the ability to block muscle wasting hormones in the body that both destroy muscle tissue and promote fat gain; as we understand, metabolic efficiency is key to any performance athlete and blocking these hormones promotes that end. If that wasnt enough it gets even better; Testosterone-Suspension actively increases natural IGF 1 hormones in the body; a very powerful naturally occurring anabolic hormone of great importance. The Downside of Testosterone-Suspension Like all testosterone forms Testosterone-Suspension does aromatize and this can lead to many unwanted adverse side-effects of an estrogenic nature such as Gynecomastia. However, the rate of aromatase with Testosterone-Suspension appears to be higher than many other forms and excess water retention can really be a problem because of this trait. For this reason aromatase inhibitors such as Arimidex and Letrozole must necessarily be part of your supplemental routine if the side-effects are to be controlled. As alluded to, Testosterone-Suspension can be very painful and administration can be very annoying at best as it must be frequent. Testosterone-Suspension is suspended in water, as is evident in its name and water based steroids are always more painful than oil based as most our commonly compounded. Further, as a water-based steroid surviving bacterium in the compound can be a large concern when purchased from many underground labs; for this reason Testosterone-Suspension must only be purchased from a human grade line. Although this will not make the compound pain free it will largely eliminate the risk of infection which is very common in black market Suspension. Application of Testosterone-Suspension As Testosterone-Suspension carries no traditional half-life in the same light as most other anabolic steroid compounds its active duration is very short lived. For this reason injections of the hormone must be daily if results are going to be seen. While daily injections will work, multiple daily injections, 2-3 per day will prove to be the most efficient and far superior to once per day. For this reason many will choose not to use the compound. However, for those who do, because Testosterone-Suspension is ester free testosterone levels will spike almost instantaneously post injection and the benefits of testosterone use will begin to show almost overnight. Testosterone Suspension Results As far as results of the cycle, one should be very happy with the results as long as the diet and training regimen are good. As previously stated, testosterone is a highly anabolic and androgenic hormone, it has an anabolic (muscle building) rating of 100, making it a good steroid to use if one is in pursuit of more size and strength. Well, lets get on with it and look at exactly what makes Testosterone Suspension a good mass builder. Firstly, testosterone promotes nitrogen retention in the muscle(2) the more nitrogen the muscles holds the more protein the muscle stores. Testosterone can also increase the levels of another anabolic hormone, IGF-1, in muscle tissue(3). Testosterone Suspension also has the amazing ability to increase the activity of satellite cells(4). These cells play a very active role in repairing damaged muscle. Testosterone also binds to the androgen receptor to promote A.R dependent mechanisms for both muscle gain as well as fat loss.(5) Testosterone significantly increases the concentrations of the A. R in cells which are critical for muscle repair and growth.(4, 6 ). Testosterone Suspension induces changes in shape and size of your muscle fibers, and also can change the actual appearance and the number of muscle fibers(7). Also of note to both bodybuilders and athletes is that many anabolic androgenic steroids (like Testosterone Suspension) can also protect your hard earned muscle from the catabolic (muscle wasting) glucocorticoid hormones(8) that your body employs to maintain homeostasis. In addition, Testosterone has the added ability to increase red blood cell production(9), and a higher RBC count may improve endurance via better oxygenated blood. More RBCs can also improve recovery from strenuous physical activity, and this has obvious benefits for the hard training bodybuilder or athlete. As with 99% of other steroids, Testosterones anabolic/androgenic effects are dose dependent, the higher the dose of Testosterone Suspension, the higher the muscle building effect(10). Testosterone Suspension Dosage Testosterone Suspension is best run for at least 6 weeks and depending on the experience of the user one may choose to supplement much longer. Since more advanced performance enhancers primarily use this hormone, other steroids are usually incorporated into the cycle. One should opt for other mass drugs such as Dianabol and Deca Durabolin since the goal of this cycle will most likely be and should be for mass. The user should expect to see rapid muscle growth, water retention, and possibly extra fat deposits. Some athletes will also choose to inject Testosterone Suspension before a workout or competition (this would increase aggression, and would be especially important for MMA competitors, or those in a sport where aggression is a benefit). Many other athletes will also use it solely for this purpose; every day (painful) shots are just not much fun for a typical 12 week cycle. It is for this reason that most people who use this steroid employ it pre-workout and/or competition, and not much more often. A mere 100mgs pre-workout or competition is sufficient, and would benefit competitive athletes greatly enough to justify its inclusion during an in-season-cycle.
  15. Sustanon 250 is a blend of four testosterone esters testosterone propionate, testosterone phenylpropionate, testosterone isocaproate and testosterone decanoate. These esters make Sustanon one of the longest-lasting steroid compounds available today. It is an ideal compound for putting on size and increasing muscle strength. Sustanon is also relatively mild on the estrogenic side effects such as gynocomastia and water-retention. Doses of 250 mgs to 1000 mgs per week are recommended to keep a balanced testosterone level, although Sustanon will stay active in the body for up to a whole month. At higher doses, estrogenic effects can be severe and anti-estrogens like Nolvadex or Proviron are recommended. Taking Sustanon will also reduce the body’s natural production of testosterone so a post-cycle therapy of HCG or Clomid is also desirable. Sustanon 250® is an oil-based injectable testosterone blend, developed by Organon. It typically contains four different testosterone esters: Testosterone propionate (30 mg); testosterone phenylpropionate (60 mg); testosterone isocaproate (60mg); and testosterone decanoate (100 mg), although a lower dosed version is also produced. An intelligently “engineered” testosterone, Sustanon is designed to provide a fast yet extended release of testosterone. The propionate and phenylpropionate esters in this product are quickly utilized, releasing into circulation within the first four days. The remaining esters are much slower to release, staying active in the body for about two and three weeks (respectively). Being a strong androgen, we can expect the typical side effects. This includes oily skin, acne body/facial hair growth and premature balding. The addition of Proscar/Propecia should be able to minimize such side effects, as it will limit the conversion of testosterone to DHT (dihydrotestosterone) . Sustanon will also suppress natural testosterone production rather quickly. The use of HCG and/or Clomid/Nolvadex are necessary at the conclusion of a cycle in order to avoid a hormonal crash. Remember though, Sustanon will remain active in the body for up to a month after your last injection was given. Beginning you post cycle drug therapy immediately after the steroid has been discontinued will not be very effective. Instead, HCG or Clomid/Nolvadex should be delayed three weeks, until you are near the point where blood androgen levels have dropped significantly. Although Sustanon remains active in the body for approximately three weeks, injections are taken at least every 10 days. An effective dosage ranges from 250mg (one ampule) a week, to 1000mg (four ampules) weekly. Some athletes do use more extreme dosages of this steroid, but this is really not a recommended practice. When the dosage rises above 750-1000mg per week, increased side effects will no doubt be outweighing additional benefits. Basically you will receive a poor return on your investment, which with Sustanon can be substantial. Instead of taking unnecessarily large amounts, athletes interested in rapid size and strength will usually opt to addition another compound. For this purpose we find that Sustanon stacks extremely well with the potent orals Anadrol and Dianabol. On the other hand, Sustanon may work better with trenbolone or Winstrol if the athlete were seeking to maintain a harder, more defined look to his physique. Sustanon 250 is probably the most sought after injectable testosterone. I must however emphasize that this is not due to an unusual potency of this testosterone combination however (remember esters only effect the release of testosterone), but simply because a “stack” of four different esters is a very good selling point. In many instances you will get a lot more for your money with enanthate, so don’t let the fancy stack fool you. Sustanon is however still very abundant on the U.S. black market, and doesn’t stay long on dealer’s shelves. In fact the high demand for this steroid has stirred new interest in its manufacture, particularly by veterinary companies in Mexico.
  16. Proviron is an oral DHT steroid compound similar to Masteron. Although it is not an ideal compound for building muscle (actually it is not good at all for this purpose), Proviron is helpful in stacks because of its unique ability to keep the body from turning testosterone into estrogen, thus giving the testosterone a better anabolic effect. This aids the bodybuilder in many ways. First, it helps reduce estrogenic side effects of other steroids water-retention, lowered sex drive, gynocomastia, etc. Also, Proviron can help boost the potency of testosterone in the body by freeing testosterone from its binding to sex hormone-binding globulin (SHBG). Proviron is therefore best stacked with testosterone, which makes taking anti-estrogen compounds unnecessary. However, Proviron can cause high blood pressure so blood pressure medication may be required for those prone to hypertension. Proviron® is the Schering brand name for the oral androgen mesterolone (1 methyl-dihydrotestosterone). Just as with DHT, the activity of this steroid is that of a strong androgen which does not aromatize into estrogen. In clinical situations Proviron is generally used to treat various types of sexual dysfunction, which often result from a low endogenous testosterone level. It can usually reverse problems of sexual disinterest and impotency, and is sometimes used to increase the sperm count. The drug does not stimulate the body to produce testosterone, but is simply an oral androgen substitute that is used to compensate for a lack of the natural male androgen. Although this steroid is strongly androgenic, the anabolic effect of it is considered too weak for muscle building purposes. This is due to the fact that Proviron is rapidly reduced to inactive metabolites in muscle tissue, a trait also characteristic of dihydrotestosterone. The belief that the weak anabolic nature of this compound indicated a tendency to block the androgen receptor in muscle tissue, thereby reducing the gains of other more potent muscle building steroids, should likewise not be taken seriously. In fact due to its extremely high affinity for plasma binding proteins such as SHBG, Proviron may actually work to increase the activity of other steroids by displacing a higher percentage into a free, unbound state. Among athletes Proviron is primarily used as an anti-estrogen. It is believed to act as an anti-aromatase in the body, preventing or slowing the conversion of steroids into estrogen. The result is somewhat comparable to Arimidex (though less profound), the drug acting to prevent the buildup of estrogen in the body. This is in direct contrast to Nolvadex, which only blocks the ability of estrogen to bind and activate receptors in certain tissues. The anti-aromatization effect is preferred, as it is a more direct and efficient means of dealing with the problem of estrogenic side effects. Another disadvantage of Nolvadex is that if discontinued too early, a rebound effect may occur as high serum estrogen levels are again free to take action. This of course could mean a rapid onset of side effects such as gynecomastia. Most actually prefer to use both Proviron and Nolvadex, especially during strongly estrogenic cycles. With each item attacking estrogen at a different angle, side effects are often greatly reduced. The anti-estrogenic properties of Proviron are not unique to this compound. A number of steroids have in fact demonstrated similar activity. Dihydrotestosterone and Masteron (2methyl-dihydrotestosterone) for example have been successfully used as therapies for gynecomastia and breast cancer due to their strong anti-estrogenic effect. It has been suggested that nandrolone may even lower aromatase activity in peripheral tissues where it is more resistant to estrogen conversion (the most active site of nandrolone aromatization seems to be the liver). The anti-estrogenic effect of all of these compounds is presumably caused by their ability to compete with other substrates for binding to the aromatase enzyme. With the aromatase enzyme bound to the steroid, yet being unable to alter it, and inhibiting effect is achieved as it is temporarily blocked from interacting with other hormones. This drug is also favored by many during contest preparations, when a lower estrogen/high androgen level is particularly sought after. This is especially beneficial when anabolics like Winstrol, oxandrolone and Primobolan are being used alone, as the androgenic content of these drugs is relatively low. Proviron can supplement a well needed androgen, and bring about an increase in the hardness and density of the muscles. Women in particular find a single 25mg tablet will efficiently shift the androgen/estrogen ratio, and can have a great impact on the physique. Since this is such a strong androgen however, extreme caution should be taken with administration. Higher dosages clearly have the potential to cause virilization symptoms quite readily. For this reason females will rarely take more than one tablet per day, and limit the length of intake to no longer than four or five weeks. One tablet used in conjunction with 10 or 20mg of Nolvadex can be even more efficient for muscle hardening, creating an environment where the body is much more inclined to burn off extra body fat (especially in female trouble areas like the hips and thighs). The typical dosage for men is one to four 25 mg per tablets per day. This is a sufficient amount to prevent gynecomastia, the drug is often used throughout the entire cycle. As mentioned earlier, it is often combined with Nolvadex (tamoxifen citrate) or Clomid (clomiphene citrate) when heavily estrogenic steroids are being taken (Dianabol, testosterone etc.). Administering 50mg of Proviron and 20mg Nolvadex daily has proven extremely effective in such instances, and it is quite uncommon for higher dosages to be required. And just as we discussed for women, the androgenic nature of this compound is greatly welcome during contest preparation. Here again Proviron should noticeably benefit the hardness and density of the muscle, while at the same time increasing the tendency to burn off a greater amount of body fat. Proviron is usually well tolerated and side effects (men) are rare with dosages under 100 mg per day. Above this, one may develop an excessively high androgen level and encounter some problems. Typical androgenic side effects include oily skin, acne, body/facial hair growth and exacerbation of a male pattern baldness condition, and may occur even with the use of a moderate dosage. With the strong effect DHT has on the reproductive system, androgenic actions may also include an extreme heightening of male libido. And as discussed earlier, Women should be careful around Proviron. It is an androgen, and as such has the potential to produce virilization symptoms quite readily. This includes, of course, a deepening of the voice, menstrual irregularities, changes in skin texture and clitoral enlargement. Proviron is also not a c17 alpha alkylated compound, an alteration commonly used with oral anabolic/androgenic steroids. Not using this structure in the case of Proviron removes the notable risk of liver toxicity we normally associate with oral drugs. It is therefore considered a “safe” oral, the user having no need to worry about serious complications with use. This steroid in fact utilizes the same 1-methylation we see present on Primobolan (methenolone), another well tolerated orally active compound. Alkylation at the one position also slows metabolism of the steroid during the first pass, although much less profoundly than 17 alpha alkylation. Likewise Proviron and Primobolan are resistant enough to breakdown to allow therapeutically beneficial blood levels to be achieved, although the overall bioavailability of these compounds is still much lower than methylated oral steroids. The popularity of Proviron amongst bodybuilders has been increasing in recent years. Many experienced bodybuilders have in fact come to swear by it, incorporating it effectively in most markedly estrogenic cycles. Due to high demand Proviron is now very easy to obtain on the black market. Most versions will be manufactured by Schering, and should cost about $1-$2 per 25 mg tab. This drug is packaged in both push-through strips and small glass vials, so do not let this alarm you. There is currently no need to worry about authenticity with this drug, as no counterfeits are known to exist. If money and availability does not prevent it, Arimidex, Femara, or Aromasin ares actually a much better choice than Proviron though. These drugs were designed specifically as an anti-aromatase, and works much more effectively than anything else we have available.
  17. Primobolan is one of those anabolic steroids which has a cult following not unlike the old original version of Masteron. Actually, as you can easily see from its anabolic:androgenic ratio below in the profile, its a pretty weak steroid but actually stronger(!) than Masteron in both regards. I dont know anyone who has run both compounds at the same dose. We are probably justified in speculating that youd probably get similar results from either of them, when you consider the fact that you are getting quite a bit less actual drug and more ester when you choose injectable Primobolan (which has the very long Enanthate ester attached to it) over Masteron (which has the very short propionate ester attached to it). In truth, I think part of the reason many Primobolan users have been disappointed is that they failed to use enough of it, for long enough. From its chemical structure and anabolic:androgenic rating, we can assume it is at least as effective as Masteron, on an equal Mg for mg basis. However, due to its ester (in the injectable version), it needs to be run for at least 12 weeks to see the full benefits from it. When you consider a measly dose of 400mgs of this stuff for 12 weeks will probably cost you around $500. Its easy to see why many people have tried to use less...and have been disappointed with their results. On the other hand, many competitive bodybuilders consider Primobolan indespensible to their pre-contest drud routine, and wouldnt consider dieting without it. Anyway...I think the comparison to Masteron (another great precontest drug) is the best one we can make, with reference to expected gains and results. I happen to be one of the few people who have used Drostanolone Enanthate (Masteron with the Enanthate ester attached) as well as Methenolone Enanthate (injectable Primobolan). I can tell you that the results from these two compounds, when ester and mg potency are the same, are in fact very similar. Effects of Primobolan Lets flesh out some of the various general effects of Primobolan, before we get into the differences between the oral and injectable versions... One study performed on sheep involved administering 100mgs of Methenolone, and electronically stimulating their lats (electronic stimulation was used because they kept falling off the chin-up bars). Anyway, when compared with the lat muscles of sheep who didnt receive Methenolone, the receiving group gained significantly more muscle mass as well as strength (1)(2). Its also has a relatively high affinity for binding to the AR, actually binding better than testosterone (3). This ability to strongly bind to the AR may be why Primobolan is such a good "fat burner." Strong AR binding has been positively correlated with lypolysis (fat-burning) (8). In addition, as this steroid can actually aid in reducing breast tumors, no ancillary products need be considered for use with Primobolan, and in fact, it may actually be a useful ancillary agent in its own right, similar to Masteron. Also, just like Masteron, Primobolan has no propensity to aromatize (convert to estrogen). Since it doesnt aromatize, alot of the side effects commonly associated with estrogen will not be of concern. This means water retention, acne, and gyno will be non-existent more or less. this lack of water retention combined with the slow and steady gains provided by Primo may help to explain why it has earned a reputation for creating quality muscle gains. This also helps to explain why it is so expensive. Although estrogenic sides are not a concern, hair loss still, remains a very real concern with Primobolan, as with many DHT-Derived steroids. Many primobolan fans always include Finasteride and Ketoconazole (shampoo) in cycles containing Primobolan. Although nobody would ever suggest to use Primobolan as a bulking agent, its been studied as an agent to halt wasting and possibly reverse many of the adverse effects of anemia. It is a shocking failure in both areas, according to some of the case studies Ive read, (5)(6) and this should come to no surprise to anyone. Anadrol reigns supreme in this area, and nobody in the athletic community would ever compare those two drugs. However, Michael Mooney and many other respected doctors who work with AIDS patients have found sufficient evidence to claim that Primobolan is an immune enhancer and as such is very useful for AIDS patients (not that the FDA cares...Primobolan is still not approved for sale in the United States). AIDS patients arent really in need of Bulking Drugs, so an immune enhancer like Primo which will add small, quality gains in muscle is perfect for them. And since we arent even going to vaguely consider the use of Primobolan as a bulking agent, clearly this leaves us with considering it primarily for use in gaining and maintaining lean tissue. Its a great choice for this purpose, and many competitors have used it very successfully to retain muscle while on a calorie reduced diet. The reason Primo is so useful for this purpose is that one of its primary functions is to help your body retain nitrogen (7) at a greatly enhanced rate. The greater your nitrogen retention is, the more muscle you will build. In the case of using primo as a pre-contest drug, this nitrogen retention will help you retain muscle and ensure that your dieting preferentially favors fat loss over muscle loss. Primobolan is a very unique steroid, as it is one of the few that comes in both an oral as well as an injectable version. I suppose Winstrol does also, but Primobolan actually has a different ester on the oral (acetate ) and injectable (Enanthate) versions. The oral version is one of the more interesting oral compounds Ive looked into. For starters, its one of the few compounds available to athletes and bodybuilders which is both oral as well as non-17-alpha-alkylation. This alteration is (as Im sure you remember from other stuff Ive written) what generally makes oral steroids survive their first pass through your liver, but also makes them Hepatoxic (Liver toxic). Well... oral Primo doesnt have this feature, so it is very mild on your liver (actually it basically isnt liver toxic at all), but also is largely destroyed by it, since 17 beta estrification and 1 alkylation is the method used to make this stuff orally available. Youll need to take a lot of this stuff for it to be effective... 100mgs/day of the oral version is a safe estimate for reasonable gains& for women, you could get away with less; perhaps 25mgs/day. Even though the acetate ester has a 2-3 day active life, your liver will do some damage to oral primo, so every day dosing will still be necessary. When men were given a 30-45mg dose of the oral version of Primo, they experienced a 15-65% decrease in gonadotropin levels (9). Remember, I said 100mgs is a good dose for gains... well, youll also reduce your gonadotropin levels considerably. I have personally never understood why people recommend either oral or injectable Primobolan as a possible bridging compound for this reason... maybe at a too-low-to-do-anything dose of 10mgs it could be used as a bridge. And forget about using injectable Primo to bridge& Hey... speaking about injectable Primo... Ive used this stuff at 200mgs/week and wasnt very impressed with it. Generally, I think injectable primo needs to be used at a dose of at least 350mgs/week (100mgs/Every other Day), and preferably at a dose of 400-600mgs/week. I happen to like running it with testosterone propionate, but for convenience I would imagine most people would run it with Testosterone Enanthate, to keep dosing times the same (shooting it twice per week, in most cases).
  18. PARABOLAN PARABOLAN In bodybuilding and also in powerlifting Parabolan has become the most desired injectable steroid compound. This is not without reason since Parabolan is truly a phenomenal, unique product. Parabolan is a strong, androgenic steroid which also has a high ana-bolic effect. Whether a novice, hard gainer, power lifter, or pro body-builder, everyone who uses Parabolan is enthusiastic about the re-sults: a fast gain in solid, high-quality muscle mass accompanied by a considerable strength increase in the basic exercises. in addition, the regular application over a number of weeks results in a well visible increased muscle hardness over the entire body without diet-ing at the same time. Frequently the following scenario takes place: bodybuilders who use steroids and for some time have been stag-nate in their development suddenly make new progress with Parabolan. Another characteristic is that Parabolan, unlike most highly-androgenic steroids, does not aromatize. The substance trenbolone does not convert into estrogens so that the athlete does not have to fight a higher estrogen level or feminization symptoms. Those who use Parabolan will also notice that there is no water retention in the tissue. To say it very clearly: Parbolan is the number one competition steroid. When a low fat content has been achieved by a low-calorie diet, Parabolan gives a dramatic increase in muscle hardness. In combination with a protein-rich diet it becomes espe-cially effective in this phase since Parabolan speeds up the metabo-lism and accelerates the burning of fat. The high androgenic effect prevents a possible overtraining syndrome, accelerates the regen-eration, and gives the muscles a full, vascular appearance but, at the same time, a ripped and shredded look. Most athletes inject Parabolan at least twice a week; some bodybuilders inject 1-2 ampules per day during the last three to four weeks be-fore a competition. Normally a dosage of 228 mg/week is used, corresponding to a weekly amount of three ampules. It is our expe-rience that good results can be achieved by injecting a 76 mg am-pule every 2-3 days. Parabolan combined with Winstrol Depot works especially well and gives the athlete a distinct gain in solid and high quality muscles together with an enormous strength gain. A very effective stack is 76 mg Parabolan every 2 days combined with 50 mg Winstrol every 2 days. Athletes who are interested in a fast mass gain often also use 30 mg Dianabol/day while those who are more interested in quality and strength like to add 25 mg+ Oxandrolone/ day. Probably the most effective Parabolan combination consists of 228 mg Parabolan/week, 200 mg Winstrol Depot/week, and 40-50 mg Oral-Turinabol/day and usually results in a drastic gain in high quality muscle mass together with a gigantic strength gain. Parabolan also seems to bring extraordinarily good results when used in combination with growth hormones. Parabolan is not a steroid suitable for year-round treatment since it is quite toxic. The duration of intake should be limited to a maxi-mum of 8 weeks. It has been proven that Parabolan, above all, puts stress on the kidneys, rather than the liver. Athletes who have taken it in high dosages over several weeks often report an unusually dark colored urine. In extreme cases blood can be excreted through the urine, a clear sign of kidney damage. Those who use Parabolan should drink an additional gallon of fluid daily since it helps flush the kidneys. Since Parabolan does not cause water and salt retention the blood pressure rarely rises. Similar to Finaject, many athletes show an aggressive attitude which is attributed to the distinct an-drogenic effect. It is interesting that acne and hair loss only occur rarely which might be due to the fact that the substance is not con-verted into dihydrotestosterone (DHT). Some athletes report nau-sea, headaches, and loss of appetite when they inject more than one ampule (76 mg) per week. Since Parabolan considerably reduces the endogenic testosterone production, the use of testosterone-stimu-lating compounds at the end of intake is suggested. In older athletes there is an increased risk that Parabolan could induce growth of the male prostate gland. We recommend that male bodybuilders, dur-ing and after a treatment with Parabolan, have their physician check their prostate to be sure it is still small in size. Steroid novices should not (yet) use Parabolan. The same is true for women; however, there are enough female athletes who do not care since the female organism reacts to the androgenic charge and the strong anabolic effect of Parabolan with distinct gains in muscles and strength, especially from a female point of view. Thus the entire body has a harder and more athletic look. Parabolan without a doubt is an enticing product for ambitious female athletes. In the end everything depends on your personal willingness to take risks, ladies. The fact is that the standards on the national and interna-tional competition scenes in female bodybuilding have achieved lev-els which cannot be reached without the administration of strongly androgenic steroid compounds. A combination well-liked by female bodybuilders consists of 76 mg Parabolan/week, 20 mg Winstrol tablets/day, and 100 mcg Clenbuterol/day Women who do not in-ject more than one ampule of Parabolan per week and who limit the period of intake to 4-5 weeks can mostly avoid or minimize virilization symptoms. Female athletes who are overdoing it or who are sensitive to the androgenic part of trenbolone hexahydrobencylcarbonate can be confronted with some unpleas-ant surprises after several weeks of use: acne, androgenically-caused hair loss on the scalp, irregular menstrual cycles, missed periods, much higher libido, aggressiveness, deep voice, chtorial hypertro-phy, and increased hair growth on face and on the legs. The last three side effects are mostly irreversible changes
  19. Masteron is a powerful anabolic/androgenic steroid derived from DHT that was designed to fight certain forms of breast cancer. It is used by bodybuilders as a bulking and cutting agent, as well as an ancillary drug to combat estrogenic side effects like water-retention. Its toxicity to the liver is very low, although side effects such as acne, hair loss and prostrate enlargement are common. Masteron is an injectable preparation containing the steroid drostanolone propionate. Drostanolone is a derivative of dihydrotestosterone, most specifically 2alpha-methyldihydrotestosterone. As a result, the structure of this steroid is that of a moderate anabolic/potent androgen which does not aromatize to estrogen. Water retention and gynecomastia therefore do not come into play with this drug. Masteron may in fact exhibit anti-estrogenic activity in the body, competing with other substrates for binding to aromatase. This would reduce the conversion rate of other steroids, Masteron acting in the same way as the oral steroid Proviron. Bodybuilders have a strong like for non-aromatizing androgens, and find Masteron very useful in a cutting phase. It is generally used for a number of weeks prior to a competition, in an effort to bring out an improved look of density and hardness to the muscles. As long as body fat percentage is low enough, Masteron should work very well. Provided everything fits as if should, the user can achieve that “ripped” look so popular to professional bodybuilding. The androgenic effect can also be crucial during this period, a time when caloric intake is drastically lowered. The user is provided added “kick” or “drive” to push through the grueling training sessions leading up to the show. Recreational users might also be interested in Masteron. Although dihydrotestosterone is not highly active in muscle tissue, the 2 alkylation present on drostanolone considerably intensifies its anabolic effect. It can therefore be used somewhat effectively as bulking agent, providing a consistent gain of high quality muscle mass. It can also be successfully combined with other steroids for an enhanced effect. Mixing drostanolone with an injectable anabolic such as Deca-Durabolin or Equipoise can prove quite useful for example, the two providing notably enhanced muscle gain without excessive water retention. For greater mass gains, a stronger androgen such as Dianabol or an injectable testosterone would do the trick. The result here can be an extreme muscle gain, with a lower level of water retention & other estrogenic side effects than if these steroids were used alone (usually in higher doses). Masteron could of course be used during cutting phases of training as well. A cycle of this drug combined with Winstrol, Primobolan or Oxandrolone should provide great muscle retention and fat loss, during a period which can be very catabolic without steroids. It is an added benefit that none of these steroids aromatize, and therefore there is no additional worry of unwanted water and fat retention. Since the propionate ester is used with this compound, injections need to be repeated at least every 3 or 4 days in order to maintain a consistent level of hormone in the blood. The weekly dosage is in the range of 300-500mg. Since estrogen is not an issue, side effects are generally mild with this steroid. As discussed earlier, gynecomastia, water retention, and high blood pressureare not a problem. Masteron is also not liver toxic, so there is little concern stress will be placed on this organ, even during longer cycles. The only real side effects would be from the basic androgenic properties of dihydrotestosterone. These includes oily skin, acne, body/facial hair growth, aggression and accelerated hair loss. Since this compound is already a synthetic DHT, Proscar would have no impact on the level of androgenic effects. Men with a receding hairline or those with a predisposition for baldness may therefore wish to stay away from Masteron completely, as the potent androgenic effect of this steroid can easily accelerate this condition.
  20. Halotestin is a good compound for use by athletes because it can greatly increase strength and energy output. Unfortunately for bodybuilders, its muscle-building attributes are not as effective. Halotestin doesn’t convert to estrogen in the body, but it is toxic to the liver, so small doses are recommended. Halotestin is the Upjohn brand name for the steroid fluoxymesterone. Structurally fluoxymesterone is a derivative of testosterone, differing from our base androgen by three structural alterations (specifically l7alpha-methyl, 11 beta-hydroxy and 9-fluoro group additions). The result is a potent oral steroid that exhibits extremely strong androgenic properties. This has a lot to due with the fact that it is derived from testosterone, and as such shares important similarities to this hormone. Most importantly, like testosterone, Halotestin appears to be a good substrate for the 5-alpha reductase enzyme. This is evidenced by the fact that a large number of its metabolites are found to be 5-alpha reduced androgens, which coupled with its outward androgenic nature, suggests it is converting to a much more active steroid in androgen responsive target tissues such as the skin, scalp and prostate. The 11 beta-hydroxyl group also inhibits aromatization, making estrogen production impossible with this steroid. Estrogenic side effects such as water retention, fat fain and gynecomastia are therefore not a concern when taking this compound. Strong androgenic side effects are to be expected though, and in many cases are unavoidable. Oily skin and acne a very common for instance, at times requiring sensitive individuals to seek some form of topical or even prescription drug treatment to keep it under control. Hair loss is an additional worry, making Halotestin a poor choice for those with an existing condition. Aggression may also become very pronounced with this drug. This effect is often desired by users looking to “harness” this in order to increase the intensity of workouts or a competition. Clearly Halotestin is a strong androgen, and definitely one female athletes should stay away from. Masculinizing side effects can be intense, and may occur very rapidly with this substance. Even women daring enough to take Dianabol should think twice about this compound, as virilization symptoms are most often permanent. Although Halotestin appears to be more androgenic than testosterone, the anabolic effect of it is not very strong. This makes it a great strength drug, but not the best for gaining serious muscle mass. The predominant effect seen when taking Halotestin is a harder, more dense look to the muscles without a notable size increase. It is therefore very useful for athletes in weight-restricted sports like wrestling, powerlifting and boxing. The strength gained from each cycle will not be accompanied by a great weight increase, allowing most competitors to stay within a specified weight range. Halotestin also makes an excellent drug for bodybuilding contest preparation. When the competitor has an acceptably low body fat percentage, the strong androgen level (in absence of excess estrogen) can elicit an extremely hard and defined (“ripped”) look to the muscles. The shift in androgen/estrogen ratio additionally seems to bring about a state in which the body may be more inclined to burn off excess fat and prevent new fat storage. The “hardening” effect of Halotestin would therefore be somewhat similar to that seen with trenbolone, although it will be without the same level of mass gain. Clearly non-aromatizing androgens such as Halotestin and trenbolone can play an important role during contest preparations. The main concern with this steroid is that it can be a very toxic drug. This is due to the fact that fluoxymesterone is a 17 alpha alkylated compound, its structure altered to survive oral administration. l7alpha alkylation can be very harsh to the liver. The possibility of damage is therefore a legitimate concern with Halotestin, especially when used at higher doses or for prolonged periods of time. The total daily dosage is likewise best kept in the range of 20-40mg, used for no longer than 8 weeks. After which an equally long break (at a minimum) should be taken from all c17-AA orals. One should also resist the temptation to stack this drug with other alkylated orals if possible, and instead opt for orals without this alteration or esterified injectable compounds (which will not add to the strain on the liver). In cutting phases a mild anabolic such as Deca-Durabolin or Equipoise might prove to be a good addition, as both provide good anabolic effect without excessive estrogen buildup. Here Halotestin will provide a well needed androgenic component, helping to promote a more solid and defined gain in muscle mass than obtained with an anabolic alone. Perhaps Primobolan Depot would even be a better choice, as with such a combination there is no buildup of estrogen (and likewise even less worry of water and fat retention). For mass we could alternately use an injectable testosterone. A mix of 400-800mg Testosterone enanthate and 20-30mg Halotestin for example, should prove to be an exceptional stack for strength and muscle gain. This however would be accompanied by a more significant level of side effects, both compounds exhibiting strong androgenic activity in the body. Fluoxymesterone also seem to depress endogenous testosterone levels rather quickly with use, despite its complete lack of estrogen conversion. One therefore should consider ancillary drug use at the conclusion of each cycle in order to help restore the normal release of androgens in the body. Using a combination of HCG and Clomid/Nolvadex is of course the best option, the two drugs working well together to restore normal hormonal functioning. Although estrogen is not a problem with Halotestin, the use of an anti-estrogen such as Nolvadex or Clomid is still indicated when discontinuing a cycle. Since HCG stimulates aromatase activity in the Leydig’s cells, here Nolvadex/Clomid help by blocking the activity of any excess estrogen that may be produced. Afterward they will also block the inhibitory effect of endogenous estrogens on the hypothalamus, stimulating the enhanced release of gonadotropins and supporting the normal biosynthesis of testosterone. Since Halotestin is only used for a few specific purposes, it is not in high demand among athletes. Likewise it is not a very popular item on the black market. Investing in the manufacture of a counterfeit version would probably not pay off well, no doubt the reason we haven’t seen any yet. All of the various forms of Halotestin could therefore be assumed legitimate when found in circulation. Currently the most popular item found on the black market is the Stenox brand from Mexico, sold in boxes of 20 tablets. Although the dosage of these tablets is only 2.5mg, the low price usually asked for this preparation more than compensates. Overall, Halotestin is an effective steroid for a narrow range of uses, and is probably not the most ideal product for the recreational user.
  21. Equipoise is a steroid compound that can give users slow but steady gains during a cycle. It is also relatively safe with very few reports of the side effects caused by testosterone conversion into estrogen. For bodybuilders, it should be used with some testosterone as Equipoise can cause sexual dysfunction. Equipoise’s long-lasting ester means it should be used for a minimum 12-week cycle. Equipoise® is the popular brand name for the veterinary injectable steroid boldenone undecylenate. It is a derivative of testosterone, which exhibits strong anabolic and moderately androgenic properties. The undecylenate ester greatly extends the activity of the drug (the undecylenate ester is only one carbon atom longer than decanoate), so that clinically injections would need to be repeated every three or four weeks. In the veterinary feild Equipoise is most commonly used on horses, exhibiting a pronounced effect on lean bodyweight, appetite and general disposition of the animal. As with all steroids, this compound shows a marked ability for increasing red blood cell production. In recent years this compound has become a favorite among athletes. Many consider it an ideal replacement to Deca-Durabolin. The side effects of Equipoise are generally mild. The structure of boldenone does allow it to convert into estrogen, but it does not have an extremely high affinity to do so. If we look at aromatization studies, they suggest that its rate of estrogen conversion should be about half that of testosterone’s. Water retention with this drug would therefore be slightly higher than that with Deca-Durabolin (with an estimated 20% conversion), but much less than we would find with a stronger compound as Testosterone. While there is still a chance of encountering an estrogen related side effect as such when using Equipoise, problems are usually not encountered at a moderate dosage level. Gynecomastia might become a problem, but usually only with very sensitive individuals or (again) with those using higher dosages. If estrogenic effects become a problem, the addition of Nolvadex should of course make the cycle more tolerable. An anti-aromatase such as Arimidex, Femara, or Amonasin would be a stronger option, however probably not necessary with such a mild drug. Although typically dosage related, Equipoise can also produce distinct androgenic side effects. Oily skin, acne, increased aggression and hair loss are all possible with this compound. Women find this drug quite comfortable, virilization symptoms usually unheard of when taken at low doses. Boldenone does reduce to a more potent androgen (dihydroboldenone) via the 5alpha reductase enzyme (which produces DHT from testosterone), however its affinity for this interaction in the human body is low to nonexistent. Therefore the reductase inhibitor Proscar would not be of much use with Equipoise, as it would be blocking what is at best an insignificant path of metabolism for the steroid. Although this drug is relatively mild, it still has a depressive effect on endogenous testosterone levels, therefore a proper post cycle therapy HCG and Clomid/Nolvadex is needed at the conclusion of each cycle to avoid a “crash”. A waiting time of around 3 weeks is required before starting PCT, enabling enough of the drug to clear one’s system to make PCT effective. In order to maintain stable blood levels, Equipoise should be injected at least once per week. It is most commonly used at a dosage of 400-600mg per week for men, 50-150 mg per week for women. Equipoise is not a rapid mass builder, but will provide a slow but steady gain of strength and quality muscle mass. The most positive effects of this drug are seen when it is used for longer cycles, usually lasting at least 10 weeks in length. The muscle gained should not be the smooth bulk seen with androgens, but instead a very defined and solid look. Since water bloat is not contributing greatly to the diameter of the muscle, much of the size gained on a cycle of Equipoise can be retained after the drug has been discontinued. It is interesting to note that structurally Equipoise and the classic bulking drug Dianabol are almost identical. In the case of Equipoise the compound uses a l7beta ester (undecylenate), while Dianabol is 17 alpha alkylated. Aside from that difference, the drugs are basically the same. Of course they act quite differently in the body, which goes to show the 17-methylation effects more than just the oral efficancy of a steroid. As discussed earlier, Equipoise is a very versatile compound. We can create a number of drug combinations with it depending on the desired result. For mass, one may want to stack it with Anadrol or an injectable testosterone. The result should be an incredible gain of muscle size and strength, without the same intensity of side effects if using the androgen (at a higher dose) alone. When used in a cutting cycle, muscle hardness and density can be greatly improved when combining Equipoise with a non-aromatizable steroid such as trenbolone acetate, Halotestin, or Winstrol. For some however, even the low buildup of estrogen associated with this compound is enough to relegate its use to bulking cycles only. Equipoise is not an ideal steroid for the drug tested athlete however. This drug has the tendency to produce detectable metabolites in the urine months after use, a worry most commonly associated with Deca-Durabolin. This is of course due to the high oil solubility of long chain esterified injectable steroids, a property which enables the drug to remain deposited in fatty tissues for extended periods of time. While this will reliably slow the release of steroid into the blood stream, it also allows small residual amounts to remain present in the body far after the initial injection. The release of stubborn stores of hormone would no doubt also be enhanced around contest time, a period when the athlete drastically attempts to mobilize unwanted body fat. If enough were used in the off-season, the athlete may actually fail a drug screen for boldenone although many months may have past since the drug was last injected.
  22. Nandrolone decanoate Deca-Durabolin; 19-Nortestoterone decanoate Molecular Formula C28H44O3 Molecular Weight 428.65 CAS Registry Number 360-70-3 EINECS 206-639-3 Melting point 33-37 ºC alpha 32 º Possibly the most popular steroid compound of the last few decades, Deca-Durabolin earns its reputation by producing large muscle gains, aiding with joint pain and improving the immune system. These benefits come from a substance that has a relatively low rate of side effects because it doesn’t convert to estrogen as much as many of its counterparts. Not that Deca is without its problems. First, Deca needs to be taken over long periods of time (cycles of 12 weeks minimum) for it to be effective. Also, Deca must be taken with testosterone because the body’s natural levels will drop. Testosterone should also be a part of a Deca cycle’s post-cycle-therapy. Deca can also cause a good deal of water retention and acne. Deca-Durabolin® is the Organon brand name for the injectable steroid nandrolone decanoate. This compound came around early in the wave of commercial steroid development, first being made available as a prescription medication in 1962. World wide “Deca” is one of the most widely used anabolic steroids. Its popularity is due to the simple fact that it exhibits many very favorable properties. Structurally nandrolone is very similar to testosterone, although it lacks a carbon atom at the 19th position (hence its other name 19-nortestosterone). The resulting structure is a steroid that exhibits much weaker androgenic properties than testosterone. Of primary interest is the fact that nandrolone will not break down to a more potent metabolite in androgen target tissues. You may remember this is a significant problem with testosterone. Although nandrolone does undergo reduction via the same (5-alpha reductase) enzyme that produces DHT from testosterone, the result in this case is dihydronandrolone. This metabolite is weaker than the parent nandroloness, and is far less likely to cause unwanted androgenic side effects. Strong occurrences of oily skin, acne, body/facial hair growth and hair loss occur very rarely. It is however possible for androgenic activity to become apparent with this as any steroid, but with nandrolone higher than normal doses are usually responsible. Nandrolone also show an extremely lower tendency for estrogen conversion. For comparison, the rate has been estimated to be only about 20% of that seen with testosterones. This is because while the liver can convert nandrolone to estradiol, in other more active sites of steroid aromatization such as adipose tissue nandrolone is far less open to this process’. Consequently estrogen related side effects are a much lower concern with this drug. An anti-estrogen is likewise rarely needed with Deca, gynecomastia only a worry among sensitive individuals. At the same time water retention is not a usual concern. This effect can occur however, but is most often related to higher dosages. The addition of Proviron and/or Nolvadex should prove sufficient enough to significantly reduce any occurrence. Clearly Deca is a very safe choice among steroids. Actually, many consider it to be the best overall steroid for a man to use when weighing the side effects and results. It should also be noted that in HIV studies, Deca has been shown not only to be effective at safely bringing up the lean body weight of patient, but also to be beneficial to the immune system. It is of note however that nandrolone is believed to have some activity as a progestin in the body. Although progesterone is a c-19 steroid, removal of this group as in 19-norprogesterone creates a hormone with greater binding affinity for its corresponding receptor. Sharing this trait, many 19-nor anabolic steroids are shown to have some affinity for the progesterone receptor as well. This can lead to some progestin-like activity in the body, and may intensify related side effects. The side effects associated with progesterone are actually quite similar to those of estrogen, including negative feedback inhibition of testosterone production, enhanced rate of fat storage and possibly gynecomastia. Many believe the progestin activity of Deca notably contributes to suppression of testosterone synthesis, which can be marked despite a low tendency for estrogen conversion. Deca is not known as a very “fast” builder. The muscle building effect of this drug is quite noticeable, but not dramatic. The slow onset and mild properties of this steroid therefore make it more suited for cycles with a longer duration. In general one can expect to gain muscle weight at about half the rate of that with an equal amount of testosterone. A cycle lasting eight to twelve weeks seems to make the most sense, expecting to elicit a slow, even gain of quality mass. Although active in the body for much longer, Deca is usually injected once or twice per week. The dosage for men is usually in the range of 300-600mg/week. If looking to be specific, it is believed that Deca will exhibit its optimal effect (best gain/side effect ratio) at around 2mg per pound of lean bodyweight/weekly. Deca is also a popular steroid among female bodybuilders. They take a much lower dosage on average than men of course, usually around 50mg weekly. Although only slightly androgenic, women are occasionally confronted with virilization symptoms when taking this compound. Should this become a concern, the shorter acting nandrolone Durabolin would be a safer option. This drug stays active for only a few days, greatly reducing the impact of androgenic buildup if withdrawal were indicated. Endogenous testosterone levels can be a concern with Deca-Durabolin, especially after long cycles. It is therefore mandatory to incorporate ancillary drugs at the conclusion of therapy. An estrogen antagonist such as Clomid or Nolvadex is therefore commonly used for a few weeks. These both provide a good level of testosterone stimulation, although they may take a couple of weeks to show the best effect. HCG injections could be added for extra reassurance, acting to rapidly restore the normal ability of the testes to respond to the resumed release of gonadotropins. For this purpose one could administer three injections of 2500-50001.U., spaced five days apart. After which point the antagonist is continued alone for a few more weeks in an effort to stabilize the production of testosterone. Remember not to begin post cycle therapy (PCT) until after Deca has been withdrawn for around three weeks. Deca stays active for quite some time so the ancillary drugs will not be able to exhibit their optimal effect when the steroid is still being released into the bloodstream. The major drawback for competitive purposes is that in many cases nandrolone metabolites will be detectable in a drug screen for up to a year (or more) after use. This is clearly due to the form of administration. Esterified compounds have a high affinity to stay stored in fatty tissues. While we can accurately estimate the time frame it will take for a given dose to enter circulation from an injection site, we cannot know for sure that 100% of the steroid will have been metabolized at any given point. Small amounts may indeed be stubborn in leaving fatty tissue, particularly after heavy, longer-term use. Some quantity of nandrolone decanoate may therefore be left to sporadically enter into the blood stream many months after use. This process may be further aggravated when dieting for a show, a time when body fat stores are being actively depleted (possibly freeing more steroid). This has no doubt been the cause for many unexpected positives on a drug screen. The fact that nandrolone has been isolated as the “hands-off” injectable for the drug tested athlete is most likely due to its popularity (and therefore common appearance on drug screens). The same risk would of course hold true for other long chain esterified injectables such as Equipoise, and Primobolan. Those not worried about drug screens are likely to find the low water retention and good effect of this drug favorable for use in pre-contest cutting stacks. A combination of Deca and Winstrol during the weeks/months leading up to a show for example, is noted to greatly enhance to look of muscularity and definition. A strong non-aromatizing androgen like Halotestin or trenbolone could be further added, providing an enhanced level of hardness and density to the muscles. Being an acceptable anabolic, Deca can also be incorporated into bulk cycles with good results. The classic Deca and Dianabol cycle has been a basic for decades, and always seems to provide excellent muscle growth. A stronger androgen such as Anadrol or testosterone could also be substituted, producing greater results. When mixed with Deca, the androgen dosage can be kept lower than if used alone, hopefully making the cycle more comfortable. Additionally one may choose to continue Deca for a number of few weeks after the androgen has been stopped. This will hopefully harden up some of the bloat produced by the androgen, giving a more quality appearance. Remember that endogenous testosterone production will not resume during Deca therapy, and ancillaries are likewise still needed.
  23. Dianabol, or D-bol, is a strong steroid compound capable of producing large gains in muscle mass. It is also one of the oldest steroid compounds created, and despite the years of improvement in steroid technology, D-bol is still commonly used. Side effects from D-bol use are moderate, although it is toxic to the liver and high doses are not recommended. Dianabol is often used by body builders and athletes to kick start muscle gains or as a bridge between cycles of other drugs in order to maintain gains. Dianabol is the old Ciba brand name for the oral steroid methandrostenolone. It is a derivative of testosterone, exhibiting strong anabolic and moderate androgenic properties. This compound was first made available in 1960, and it quickly became the most favored and widely used anabolic steroid in all forms of athletics. This is likely due to the fact that it is both easy to use and extremely effective. In the U.S. Dianabol production had meteoric history, exploding for quite some time, then quickly dropping out of sight. Many were nervous in the late 80′s when the last of the U.S. generics were removed from pharmacy shelves, the medical community finding no legitimate use for the drug anymore. But the fact that Dianabol has been off the U.S. market for over 10 years now has not cut its popularity. It remains the most commonly used black market oral steroid in the U.S. As long as there are countries manufacturing this steroid, it will probably remain so. Similar to testosterone and Anadrol 50, Dianabol is a potent steroid, but also one which brings about noticeable side effects. For starters methandrostenolone is quite estrogenic. Gynecomastia is often a concern during treatment, and may present itself quite early into a cycle (particularly when higher doses are used). At the same time water retention can become a pronounced problem, causing a notable loss of muscle definition as both subcutaneous water and fat build. Sensitive individuals may therefore want to keep the estrogen under control with the addition of an anti-estrogen such as Nolvadex and/or Proviron. The stronger drugs Arimidex, Femara, or Aromasin (antiaromatase) would be a better choice if available. In addition, androgenic side effects are common with this substance, and may include bouts of oily skin, acne and body/facial hair growth. Aggression may also be increased with a potent steroid such as this, so it would be wise not to let your disposition change for the worse during a cycle. With Dianabol there is also the possibility of aggravating a male pattern baldness condition. Sensitive individuals may therefore wish to avoid this drug and opt for a milder anabolic such as Deca-Durabolin. While Dianabol does convert to a more potent steroid via interaction with the 5-alpha reductase anzyme (the same enzyme responsible for converting testosterone to dihydrotestosterone), it has extremely little affinity to do so in the human body’s. The androgenic metabolite 5alpha dihydromethandrostenolone is therefore produced only in trace amounts at best. Therefore the use of Proscar/Propecia would serve no real purpose. Being moderately androgenic, Dianabol is really only a popular steroid with men. When used by women, strong virilization symptoms are of course a possible result. Some do however experiment with it, and find low doses (5mg) of this steroid extremely powerful for new muscle growth. Whenever taken, Dianabol will produce exceptional mass and strength gains. It’s effectiveness is often compared to other strong steroids like testosterone and Anadrol 50, and it is likewise a popular choice for bulking purposes. A daily dosage of 20-40mg is enough to give almost anybody dramatic results. Some do venture much higher in dosage, but this practice usually leads to a more profound incidence of side effects. It additionally combines well with a number of other steroids. It is noted to mix particularly well with the mild anabolic Deca-Durabolin. Together one can expect an exceptional muscle and strength gains, with side effects not much worse than one would expect from Dianabol alone. For all out mass, a long acting testosterone ester like enanthate can be used. With the similarly high estrogenic/androgenic properties of this androgen, side effects may be extreme with such a combination however. Gains would be great as well, which usually makes such an endeavor worthwhile to the user. As discussed earlier, ancillary drugs can be added to reduce the side effects associated with this kind of cycle. In order to withstand oral administration, this compound is c17 alpha alkylated. We know that this alteration protects the drug from being deactivation by the liver (allowing nearly all of the drug entry into the bloodstream), however it can also be toxic to this organ. Prolonged exposure to c17 alpha alkylated substances can result in actual damage, possibly even the development of certain kinds of cancer. To be safe one might want to visit the doctor a couple of times during each cycle to keep an eye on their liver enzyme values. Cycles should also be kept short, usually less than 8 weeks long to avoid doing any noticeable damage. Jaundice (bile duct obstruction) is usually the first visible sign of liver trouble, and should be looked out for. This condition produces an unusual yellowing of the skin, as the body has trouble processing bilirubin. In addition to the skin, the whites of the eyes may also yellow, a clear indicator of trouble. Should this occur the drug should be discontinued immediately and a doctor visited. This is usually a point where further, permanent damage can be avoided. It is also interesting to note that methandrostenolone is structurally identical to boldenone (EQ), except that it contains the added c17 alpha alkyl group discussed above. This fact makes clear the impact of altering a steroid in such a way, as these two compounds appear to act very differently in the body. The main dissimilarity seems to lie in the tendency for estrogenic side effects, which seems to be much more pronounced with Dianabol. Equipoise is known to be quite mild in this way, and users therefore commonly take this drug without any need of an anti-estrogen. Dianabol is much more estrogenic not because it is more easily aromatized, as in fact the 17 alpha methyl group and c1-2 double bond both slow the process of aromatization. The problem is that methandrostenolone converts to l7alpha methylestradiol, a more biologically active form of estrogen than regular estradiol. But Dianabol also appears to be much more potent in terms of muscle mass compared to boldenone, supporting the notion that estrogen does play an important role in anabolism. In fact boldenone and methandrostenolone differ so much in their potencies as anabolics that the two are rarely though of as related. As a result, the use of Dianabol is typically restricted to bulking phases of training while Equipoise is considered an excellent cutting or lean-mass building steroid. The half-life of Dianabol is only about 3 to 4 hours, a relatively short time. This means that a single daily dosage schedule will produce a varying blood level, with ups and downs throughout the day. The user likewise has a choice, to either split up the tablets during the day or to take them all at one time. The usual recommendation has been to divide them and try to regulate the concentration in your blood. This however, will produce a lower peak blood level than if the tablets were taken all at once, so there may be a trade off with this option. The steroid researcher Bill Roberts also points out that a single-episode dosing schedule should have a less dramatic impact on the hypothalamic-pituitary-testicular axis, as there is a sufficient period each day where steroid hormone levels are not extremely exaggerated. I tend to doubt hormonal stability can be maintained during such a cycle however, but do notice that anecdotal evidence often still supports single daily doses to be better for overall results. Perhaps this is the better option. Since we know the blood concentration will peak about 1.5 to 3 hours after administration, we may further wonder the best time to take our tablets. It seems logical that taking the pills earlier in the day, preferably some time before training, would be optimal. This would allow a considerable number of daytime hours for an androgen rich metabolism to heighten the uptake of nutrients, especially the critical hours following training.
  24. Testosterone undecanoate Andriol; 17-[(1-Oxoundecyl)oxy]-androst-4-en-3-one Molecular Formula C30H48O3 Molecular Weight 456.70 CAS Registry Number 5949-44-0 EINECS 227-712-6 Andriol is an oral steroid that produces mild gains and extremely mild unwanted side effects. Unfortunately, it is also an expensive steroid and to make it worthwhile for athletes and bodybuilders to see results from its use, a lot needs to be taken. Andriol is a unique oral testosterone product, developed by the international drug firm Organon. One of the more recently developed anabolic steroids, Andriol first became available in the early 1980′s. This compound contains 40 mg of testosterone undecanoate, based in oil (oleic acid) and sealed inside a capsule. Subtracting the ester weight, this equates to a dosage of approximately 25mg of raw testosterone per cap. The design of this steroid is quite different from that of most oral steroids. Drugs administered orally generally enter the blood stream through the liver. When a steroid compound is given this way without some form of structural protection, it will be quickly broken down during the “first pass”. This process leaves very little steroid intact, basically deactivating the drug. Adding a methyl group (c-17 AA) to the structure is one way to protect it from this process, however stress is also placed on the liver as a result. In some instances this stress can lead to actual damage to liver tissues, so the designers of this steroid sought another way to protect the testosterone molecule. With Andriol, this was accomplished by making a form of testosterone that would be absorbed through the lymphatic system. This is due to its high fat solubility brought about by the ester, and its suspension in oil. Having the compound absorbed this way was thought to be very advantageous, as it allows the steroid to bypass the destructive first-pass through liver. This should permit the compound to enter the blood stream intact, without the need for a harsh chemical alteration. The ester breaks off once it is in circulation of course, yielding free active Pharmacokinetics of Oral Testosterone. In design this steroid appears to be undecanoate that of a completely liver safe and orally active form of testosterone. On paper this drug seems like a great oral testosterone product. Clean, safe and worlds apart from other oral testosterone derivatives like the crude methyltestosterone. But as we always hear in life, if it looks to good to be true, it probably is. There are definitely some issues with Andriol. The first problem is that bioavailability, although clearly worlds apart from trying to take straight testosterone orally, is probably not significant next to c17alpha alkylated orals. Athletes typically find that in doses of less than 240mg per day (6 capsules) effects are generally not seen at all. 240mg of testosterone ester daily, the primary male androgen, and only a meager effect. When doses go higher, maybe 8-10 capsules (320-400mg), new muscle growth is slight to moderate at best, but no incredible bulky gains are ever reported. Logic leads one to believe that only a little testosterone is making its way into circulation. Testosterone is a powerful hormone no matter what the ester or form of administration. If it were active in the blood stream, the results would have to be pronounced. When one injects an oil based testosterone ester like cypionate, a dosage of 400mg per week is more than sufficient to see results. 400mg Andriol per day should be packing on an incredible amount of mass. Where does it all go? Individual problems with absorption may play a role into things here. Clearly there is little to be said except that this drug is unpredictable in its ability to be absorbed and utilized by the body. While one day you might be getting great absorption, perhaps the next day you are getting very little. Studies with men were no better than with women, where again this drug was shown to be unpredictably absorbed and utilized with blood levels ranging from 11.5 to 60.1 nmol/L with 80mg twice daily. One might also pay interest to the “mildness” of this compound as described by other bodybuilding materials. Andriol is often spoken about as some type of magic product, which to spite being a form of regular testosterone somehow allows for only minimal estrogen conversion. You should know that the way a drug is administered includes a number of factors that can slightly alter its effect, the most predominant being the speed of release. This effects the time it takes for a peak blood level to be reached, and likely the length it takes to see results. The primary reason Testosterone suspension seems more powerful than enanthate is because more drug is active on day one. At the same time estrogen builds up faster and side effects become pronounced very quickly. The ester is also part of the total weight, and 100mg testosterone contains a much larger quantity of testosterone molecules that testosterone plus ester, another reason for varying effect. But these changes do not amount to all that much. The structure of testosterone is what allows it to break down into estrogen. The only way we can really prevent an androgen from converting to estrogen is to change the base molecule, not the ester. Once free in the blood stream we cannot prevent testosterone from being aromatized without interfering with the aromatase enzyme itself. The lack of results and side effects often reported with Andriol must be going hand in hand with poor absorption. Most athletes today consider Andriol a very poor buy. I know other references do find use for this drug, which is defendable because some amount of steroid clearly does enter the blood stream in tact. Technically it is still an oral testosterone, and definitely does not carry the same liver-toxicity risks associated with most steroids designed for this type of administration. Those specifically looking for a mild oral at times do purchase this product, and occasionally are even satisfied with their results. But for most its high price and required high daily dosages usually causes them to avoided it when crossing it on the black market. Besides, if we want a mild steroid the last thing we really should shop for is a testosterone.
  25. Oxymetholone Anasterone; 17b-Hydroxy-2-hydroxymethylene-17a-methyl-3-androstanone; 4,5-Dihydro-2-hydroxymethylene-17-a-methyltestosterone Molecular Formula C21H32O3 Molecular Weight 332.48 CAS Registry Number 434-07-1 EINECS 207-098-6 Melting point 172-180 ºC alpha 34 º Water solubility <0.1 g/100 mL at 23 ºC Anadrol 50, also referred to as A50, is a powerful steroid that produces very noticeable weight gains in a very short time. Unfortunately, it is also highly toxic in the liver and produces some very unfavorable side effects, such as headaches, and bloating. The gains from taking Anadrol 50 are very dramatic, but they tend to taper off quickly, which is why it is often stacked at the beginning of a cycle as a kick-start to fast gains. Anadrol 50® is the U.S. brand name for oxymetholone, a very potent oral androgen. This compound was first made available in 1960, by the international drug firm Syntex. Since oxymetholone is quite reliable in its ability to increase red blood cell production (and effect characteristic of most anabolic/androgenic steroids), it showed great promise in treating cases of severe anemia. It turned out to be well suited for this purpose, and was popular for quite some time. But recent years have brought fourth a number of new treatments, most notably the non-steroidal hormone Epogen (erythropoietin). This drug is shown to have a much more direct effect on the red blood cell count, without the side effects of a strong androgen. Syntex stopped in the U.S. in 1993, which was around the same time they decided to drop this item in a number of foreign countries as well. Plenastril from Switzerland and Austria was dropped; following soon was Oxitosona from Spain. Many Athletes feared Anadrol 50 might be on the way out for good. But new HIV/AIDS studies have shown a new light on oxymetholone. These studies are finding (big surprise) exceptional anti-wasting properties to the compound and believe it can be used safely in many such cases. Interest has been peaked, and as of 1998 Anadrol 50 is again being sold in the United States. This time we see the same Anadrol 50 brand name, but the manufacturer is the drug firm Unimed. Syntex continues to market & license this drug in a number of countries however (under a few different brand names). Anadrol 50 is considered by many to be the most powerful steroid available, with results of this compound being extremely dramatic. A steroid novice experimenting with oxymetholone is likely to gain 20 to 30 pounds of massive bulk, and it can often be accomplished in less than 6 weeks, with only 50-100mg a day. This steroid produces a lot of trouble with water retention, so let there be little doubt that much of this gain is simply bloat. But for the user this is often little consequence, feeling bigger and stronger on Anadrol 50 than any steroid they are likely to cross. Although the smooth look that results from water retention is often not attractive, it can aid quite a bit to the level of size and strength gained. The muscle is fuller, will contract better and is provided a level of protection in the form of “lubrication” to the joints as some of this extra water is held into and around connective tissues. This will allow for more elasticity, and will hopefully decrease the chance for injury when lifting heavy. It should be noted however, that on the other hand the very rapid gain in mass might place too much stress on your connective tissues for this to compensate. The tearing of pectoral and biceps tissue is commonly associated with heavy lifting while massing up on heavy androgens. There is such a thing as gaining too fast. Pronounced estrogen trouble also puts the user at risk for developing gynecomastia. Individuals sensitive to the effects of estrogen, or looking to retain a more quality look, will therefore often add Nolvadex to each cycle. It is important to note however, that this drug does not directly convert to estrogen in the body. Oxymetholone is a derivative of dihydrotestosterone, which gives it a structure that cannot be aromatized. As such, many have speculated as to what makes this hormone so troublesome in terms of estrogenic side effects. Some have suggested that it has progestational activity, similar to nandrolone, and is not actually estrogenic at all. Since the obvious side effects of both estrogens and progestins are very similar, this explanation might be a plausible one. However we do find medical studies looking at this possibility. One such tested the progestational activity of various steroids including nandrolone, norethandrolone, methandrostenolone, testosterone and oxymetholone. It reported no significant progestational effect inherent in oxymetholone or methandrostenolone, slight activity with testosterone and strong progestational effect inherent in nandrolone and norethandrolone. With such findings it starts to seem much more likely that oxymetholone can intrinsically activate the estrogen receptor itself, similar to but more profoundly than the estrogenic androgen methAndriol. If this is the case we can only combat the estrogenic side effects of oxymetholone with estrogen receptor antagonists such as Nolvadex or Clomid, and not with an aromatase inhibitor. The strong anti-aromatase compounds such as Arimidex, Femara, or Aromasin would prove to be totally useless with this steroid, as aromatase is not involved. Anadrol 50 is also a very potent androgen. This factor tends to produce many pronounced, unwanted androgenic side effects. Oily skin, acne and body/facial hair growth can be seen very quickly with this drug. Many individuals respond with severe acne, often requiring medication to keep it under control. Some of these individuals find that Accutaine works well, which is a strong prescription drug that acts on the sebaceous glands to reduce the release of oils. Those with a predisposition for male pattern baldness may want to stay away from Anadrol 50 completely, as this is certainly a possible side effect during therapy. And while some very adventurous female athletes do experiment with this compound, it is much too androgenic to recommend. Irreversible virilization symptoms can be the result and may occur very quickly, possibly before you have a chance to take action. It is interesting to note that Anadrol 50 does exhibit some tendency to convert to dihydrotestosterone, although this does not occur via the 5-alpha reductase enzyme (responsible for altering testosterone to form DHT) as it is already a dihydrotestosterone based steroid. Aside from the added c-17 alpha alkylation, oxymetholone differs from DHT only by the addition of a 2-hydroxymethylene group. This grouping can be removed metabolically however, reducing oxymetholone to the potent androgen l7alpha-methyl dihydrotestosterone (mesterolone; methyldihydrotestosterone). There is little doubt that this biotransformation contributes at least at some level to the androgenic nature of this steroid, especially when we note that in its initial state Anadrol 50 has a notably low binding affinity for the androgen receptor. So although we have the option of using the reductase inhibitor finasteride (Proscar) to reduce the androgenic nature of testosterone, it would be of no benefit with Anadrol 50 as this enzyme is not involved. The principle drawback to Anadrol 50 is that it is a 17alpha alkylated compound. Although this design gives it the ability to withstand oral administration, it can be very stressful to the liver. Anadrol 50 is particularly dubious because we require such a high milligram amount per dosage. The difference is great when comparing it to other oral steroids like Dianabol or Winstrol, which have the same chemical alteration. Since they have a slightly higher affinity for the androgen receptor, they are effective in much smaller doses. Anadrol 50 has a lower affinity, which may be why we have a 50mg tablet dosage. When looking at the medical requirements, the recommended dosage for all ages has been 1 – 5 mg/kg of body weight. This would give a 220lb person a dosage as high as 10 Anadrol 50 tablets (500mg) per day. There should be little wonder why when liver cancer has been linked to steroid use, Anadrol 50 is generally the culprit. Athletes actually never need such a high dosage and will take in the range of only 1-3 tablets per day. Many happily find that one tablet is all they need for exceptional results, and avoid higher amounts. Cautious users will also limit the intake of this compound to no longer than 4-6 weeks and have their liver enzymes checked regularly with a doctor. Kidney functions may also need to be looked after during longer use, as water retention/high blood pressure can take a toll on the body. Before starting a cycle, one should know to give Anadrol 50 the respect it is due. It is a very powerful drug, but not always a friendly one. When discontinuing Anadrol 50, the crash can be equally powerful. To begin with, the level of water retention will quickly diminish, dropping the user’s body weight dramatically. This should be expected, and not of much concern. What is of great concern is restoring endogenous testosterone production. Anadrol 50 will quickly and effectively lower natural levels during a cycle, so HCG and Clomid/Nolvadex are a must when discontinuing a cycle. The old practice of slowly tapering off your dosage is totally ineffective at raising testosterone levels. Without ancillary drugs, run away cortisol levels will likely strip much of the muscle that was gained during the cycle. If HCG and Clomid/Nolvadex are used properly, the person should be able to maintain a considerable amount of new muscle mass. Before going off, some alternately choose to first switch over to a milder injectable like Deca-Durabolin. This is in an effort to harden up the new mass, and can prove to be an effective practice. Although a drop of weight due to water loss is likely when making the switch, the end result should be the retention of more (quality) muscle mass with a less pronounced crash. Remember ancillaries though, as testosterone production will not be rebounding during Deca therapy.
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